SCHEMBL6449254

SCHEMBL6449254

C=CCCOC(=O)NCC(C(=O)NCCC#N)c1ccc(O)cc1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.33
CTSK P43235 3/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31
HRH4 Q9H3N8 2/20 0.31
HRH3 Q9Y5N1 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443607 0.91 CTSS (0.38) CTSSCTSKCTSLCTSB
SCHEMBL6443482 0.89 CTSS (0.44) CTSSCTSKCTSLCTSBESR1
SCHEMBL6445250 0.85 CTSS (0.35) CTSSCTSKCTSLCTSB
SCHEMBL6442609 0.85 CTSS (0.37) CTSSCTSKCTSLCTSBESR1
SCHEMBL6446503 0.84 SMN1; SMN2 (0.43) CTSSCTSKCTSLCTSBESR1
SCHEMBL6448170 0.84 CTSK (0.42) CTSSCTSKCTSLCTSBESR1
SCHEMBL6442192 0.84 ESR1 (0.40) CTSSCTSKCTSLCTSBESR1
SCHEMBL6446330 0.82 SMN1; SMN2 (0.48) ESR1
SCHEMBL6446763 0.82 ESR1 (0.41) CTSSCTSKCTSLCTSBESR1
SCHEMBL6443579 0.81 CTSS (0.38) CTSSCTSKCTSLESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed