SCHEMBL6442192

SCHEMBL6442192

CCOC(=O)NCC(C(=O)NCCC#N)c1ccc(O)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.40
ESR2 Q92731 2/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CTSS P25774 6/20 0.39
CTSK P43235 3/20 0.39
MIF P14174 2/20 0.36
CTSL P07711 3/20 0.35
CTSB P07858 2/20 0.35
LMNA P02545 1/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
POLB P06746 2/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
GLA P06280 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6442434 0.89 POLB (0.45) CTSSCTSKCTSLCTSBLMNA
SCHEMBL6442609 0.89 CTSS (0.37) ESR1ESR2CA12CA1CA2
SCHEMBL6822170 0.89 CTSS (0.49) ESR1ESR2CA12CA1CA2
SCHEMBL6446763 0.89 ESR1 (0.41) ESR1ESR2CA12CA1CA2
SCHEMBL6446503 0.89 SMN1; SMN2 (0.43) ESR1ESR2CTSSCTSKCTSL
SCHEMBL6448170 0.89 CTSK (0.42) ESR1ESR2CTSSCTSKCTSL
SCHEMBL6446330 0.87 SMN1; SMN2 (0.48) ESR1LMNASMN1; SMN2NPC1
SCHEMBL6819019 0.85 CTSS (0.48) CTSSCTSKCTSLCTSB
SCHEMBL6449254 0.84 CTSS (0.33) ESR1ESR2CTSSCTSKCTSL
SCHEMBL6443381 0.84 CYP2D6 (0.40) CTSSCTSKCTSLCTSBPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed