SCHEMBL6449437

SCHEMBL6449437

CC(C)[C@H](N)C(=O)N(C(=O)OCc1ccccn1)[C@@H](Cc1ccccc1)[C@@H](O)[C@@H](O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.44
KLK5 Q9Y337 2/20 0.43
REN P00797 12/20 0.40
PSEN1 P49768 3/20 0.39
PSEN2 P49810 3/20 0.39
APH1B Q8WW43 3/20 0.39
NCSTN Q92542 3/20 0.39
APH1A Q96BI3 3/20 0.39
PSENEN Q9NZ42 3/20 0.39
APP P05067 1/20 0.39
CTSD P07339 1/20 0.38
CTSE P14091 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9741355 1.00 CA2 (0.44) CA2KLK5RENPSEN1PSEN2
SCHEMBL6445021 0.88 PGR (0.46) CA2
SCHEMBL6449059 0.88 PGR (0.46) CA2
SCHEMBL6447678 0.88 PGR (0.46) CA2
SCHEMBL6446457 0.88 KLK5 (0.43) KLK5RENPSEN1PSEN2APH1B
SCHEMBL7275895 0.87 PGR (0.47) CA2
SCHEMBL8331514 0.85 UGT1A1 (0.41) CA2KLK5RENPSEN1PSEN2
SCHEMBL7270127 0.83 CA2 (0.53) CA2RENCTSD
SCHEMBL7334217 0.81 UGT1A1 (0.41) CA2KLK5PSEN1PSEN2APH1B
SCHEMBL7329645 0.80 UGT1A1 (0.38) CA2KLK5PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0839798-B1 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LAB (US) 2005-08-17 EP disclosed
EP-0839798-A2 Intermediates for preparating non-peptide retroviral protease inhibitors ABBOTT LABORATORIES (US) 1998-05-06 EP disclosed
US-5670675-A Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1997-09-23 US disclosed
US-5545750-A TREATING HUMAN IMMUNODEFICIENCY VIRUS ABBOTT LABORATORIES (US) 1996-08-13 US disclosed
EP-0402646-A1 Retroviral protease inhibiting compounds ABBOTT LABORATORIES (US) 1990-12-19 EP disclosed