SCHEMBL7329645

SCHEMBL7329645

COc1ccccc1CN(C[C@H](O)[C@H](Cc1ccccc1)N(C(=O)OCc1ccccn1)C(=O)[C@@H](N)C(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
UGT1A1 P22309 3/20 0.38
MLNR O43193 1/20 0.38
NR1I2 O75469 1/20 0.38
SLCO2B1 O94956 1/20 0.38
ABCB11 O95342 1/20 0.38
ABCB1 P08183 1/20 0.38
CCKAR P32238 1/20 0.38
OPRK1 P41145 1/20 0.38
GHSR Q92847 1/20 0.38
SLCO1B3 Q9NPD5 1/20 0.38
ABCG2 Q9UNQ0 1/20 0.38
SLCO1B1 Q9Y6L6 1/20 0.38
KCNH2 Q12809 1/20 0.38
ITGA4 P13612 1/20 0.38
ITGB7 P26010 1/20 0.38
SLC1A5 Q15758 1/20 0.36
KLK5 Q9Y337 1/20 0.35
PSEN1 P49768 10/20 0.35
PSEN2 P49810 10/20 0.35
APH1B Q8WW43 10/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8331514 0.93 UGT1A1 (0.41) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL7334217 0.91 UGT1A1 (0.41) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL7333582 0.87 UGT1A1 (0.36) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL8842808 0.85 SLC1A5 (0.36) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL7331827 0.82 CYP3A4 (0.41) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL8330458 0.81 CYP3A4 (0.38) UGT1A1MLNRNR1I2SLCO2B1ABCB11
SCHEMBL7336658 0.80 PGR (0.41) UGT1A1ABCB1KCNH2SLC1A5LNPEP
SCHEMBL6449437 0.80 CA2 (0.44) KLK5PSEN1PSEN2APH1BNCSTN
SCHEMBL9741355 0.80 CA2 (0.44) KLK5PSEN1PSEN2APH1BNCSTN
SCHEMBL7275895 0.79 PGR (0.47) ABCB1SLC1A5CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5990135-A FOR TREATING A RETROVIRAL INFECTION SUCH AS HIV INFECTION; FOR EXAMPLE 5S-N-((2-PYRIDINYL)METHOXYCARBONYL)VALINYLAMINO-2-((N-3 -PYRIDINYL)METHOXYCARBONYL)AMINO-4S-HYDROXY-1,6-DIPHENYL-2-AZAHEXANE AND OTHER COMPOUNDS OF GIVEN FORMULA ABBOTT LABORATORIES (US) 1999-11-23 US disclosed
US-5621109-A OXAZOLE/THIAZOLE DERIVATIVES OF HYDROXYMETHYL HYDRAZONES; SIDE EFFECT REDUCTION ABBOTT LABORATORIES (US) 1997-04-15 US disclosed
US-5461067-A For HIV infections ABBOTT LABORATORIES (US) 1995-10-24 US disclosed
WO-1994019332-A1 RETROVIRAL PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1994-09-01 WO disclosed