SCHEMBL6450360

SCHEMBL6450360

COc1ccc(CN(Cc2ccc(OC)cc2)c2nc3[nH]cnc3c(=O)[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
QTRT1 Q9BXR0 1/20 0.42
QPCT Q16769 2/20 0.42
LIG1 P18858 1/20 0.41
MAPT P10636 2/20 0.39
LMNA P02545 2/20 0.39
ALDH1A1 P00352 3/20 0.39
HPGD P15428 1/20 0.39
XDH P47989 1/20 0.39
DAO P14920 1/20 0.37
ADORA3 P0DMS8 2/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CHRM2 P08172 1/20 0.36
CYP3A4 P08684 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
DRD1 P21728 1/20 0.36
HTR2A P28223 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL251127 0.75 PIK3CA (0.44) QPCTMAPTLMNAALDH1A1MEN1
SCHEMBL155447 0.72 PDPK1 (0.41) MAPTLMNAALDH1A1HPGDMEN1
Hydrochloric Acid SCHEMBL17186359 0.70 PDPK1 (0.40) MAPTLMNAALDH1A1HPGDMEN1
Hydrochloric Acid SCHEMBL17186229 0.70 PDPK1 (0.40) MAPTLMNAALDH1A1HPGDMEN1
SCHEMBL22524079 0.70 ALDH1A1 (0.36) ALDH1A1XDHDAOADORA3CYP1A2
SCHEMBL31226407 0.69 QPCT (0.40) QPCTMAPTLMNAALDH1A1HPGD
SCHEMBL26529868 0.68 LMNA (0.64) MAPTLMNAALDH1A1HPGDMEN1
SCHEMBL31146869 0.68 QPCT (0.48) QTRT1QPCTMAPTLMNAALDH1A1
SCHEMBL17144480 0.68 SLC2A1 (0.47) QPCTMAPTLMNAALDH1A1MEN1
SCHEMBL5196594 0.67 KDM4E (0.41) QTRT1LIG1MAPTLMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539783-A1 INHIBITORS OF NUCLEOSIDE PHOSPHORYLASES AND NUCLEOSIDASES ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2005-06-15 EP disclosed
WO-2004018496-A1 INHIBITORS OF NUCLEOSIDE PHOSPHORYLASES AND NUCLEOSIDASES ALBERT EINSTEIN COLLEGE OF MEDICINE OF YESHIVA UNIVERSITY (US) 2004-03-04 WO disclosed