SCHEMBL6450858

SCHEMBL6450858

CC(=O)c1ccc(-c2ccc(-c3csc(C(=O)NCC4CCCCC4)c3)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.57
HDAC4 P56524 2/20 0.57
MMP12 P39900 4/20 0.55
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
MMP13 P45452 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC1 Q13547 1/20 0.46
MLYCD O95822 1/20 0.45
CA2 P00918 1/20 0.44
MAPK14 Q16539 4/20 0.44
TDP1 Q9NUW8 1/20 0.44
ROCK2 O75116 1/20 0.43
ROCK1 Q13464 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6452267 0.88 MMP12 (0.68) HDAC6HDAC4MMP12HDAC3HDAC1
SCHEMBL6874296 0.88 MMP12 (0.68) HDAC6HDAC4MMP12HDAC3HDAC1
SCHEMBL6457597 0.86 HDAC4 (0.56) HDAC6HDAC4MMP12MEN1KMT2A
SCHEMBL6878595 0.83 MMP12 (0.55) HDAC6HDAC4MMP12MEN1KMT2A
SCHEMBL6878598 0.83 MMP12 (0.55) HDAC6HDAC4MMP12MEN1KMT2A
SCHEMBL6371105 0.80 MMP12 (0.80) HDAC6HDAC4MMP12MEN1KMT2A
SCHEMBL6451716 0.79 MMP12 (0.81) HDAC6HDAC4MMP12MMP13HDAC3
SCHEMBL8340443 0.77 MMP12 (0.55) HDAC6HDAC4MMP12MMP13MAPK14
SCHEMBL6456462 0.74 MMP12 (0.72) HDAC6HDAC4MMP12MEN1KMT2A
SCHEMBL6455095 0.74 MMP12 (0.71) HDAC6HDAC4MMP12MMP13HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534700-A1 NOVEL THIOPHENE DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME WARNER-LAMBERT COMPANY LLC (US) 2005-06-01 EP disclosed
WO-2004018448-A1 NOVEL THIOPHENE DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME WARNER-LAMBERT COMPANY LLC (US) 2004-03-04 WO disclosed