SCHEMBL6457597

SCHEMBL6457597

O=C(NCC1CCCCC1)c1cc(-c2ccc(-c3ccncc3)cc2)cs1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 3/20 0.56
HDAC6 Q9UBN7 3/20 0.56
MMP12 P39900 5/20 0.54
ROCK2 O75116 5/20 0.52
ROCK1 Q13464 1/20 0.52
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
MMP13 P45452 2/20 0.47
MMP3 P08254 1/20 0.47
MMP9 P14780 1/20 0.47
MMP8 P22894 1/20 0.47
HDAC3 O15379 2/20 0.47
HDAC1 Q13547 1/20 0.47
PLK4 O00444 1/20 0.46
PDPK1 O15530 1/20 0.46
DAPK3 O43293 1/20 0.46
PRKD3 O94806 1/20 0.46
MAP4K4 O95819 1/20 0.46
CHEK2 O96017 1/20 0.46
CDK1 P06493 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8340443 0.88 MMP12 (0.55) HDAC4HDAC6MMP12ROCK2ROCK1
SCHEMBL6455095 0.87 MMP12 (0.71) HDAC4HDAC6MMP12ROCK2MMP13
Hydrochloric Acid SCHEMBL6881474 0.86 MMP12 (0.70) HDAC4HDAC6MMP12ROCK2MMP13
SCHEMBL6450858 0.86 HDAC6 (0.57) HDAC4HDAC6MMP12ROCK2ROCK1
SCHEMBL6882247 0.82 MMP12 (0.56) HDAC4HDAC6MMP12ROCK2MEN1
SCHEMBL6451716 0.81 MMP12 (0.81) HDAC4HDAC6MMP12MMP13MMP8
SCHEMBL26856930 0.77 PIK3CG (0.47) HDAC4HDAC6MMP12MEN1KMT2A
SCHEMBL6456462 0.76 MMP12 (0.72) HDAC4HDAC6MMP12MEN1KMT2A
SCHEMBL26856937 0.76 PIK3CG (0.48) HDAC4HDAC6MMP12HDAC3HDAC1
SCHEMBL6463535 0.75 MMP12 (0.88) HDAC4HDAC6MMP12MMP13MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534700-A1 NOVEL THIOPHENE DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME WARNER-LAMBERT COMPANY LLC (US) 2005-06-01 EP claimed
WO-2004018448-A1 NOVEL THIOPHENE DERIVATIVES, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME WARNER-LAMBERT COMPANY LLC (US) 2004-03-04 WO claimed