SCHEMBL6451847

SCHEMBL6451847

CCc1ccccc1CNC(=O)c1c(C)c(-c2ccccc2)nc2cc(OC)ccc12

nearest known ligand 0.55

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
TACR3 P29371 3/20 0.54
HPGD P15428 1/20 0.52
PTGFR P43088 11/20 0.52
LMNA P02545 2/20 0.49
TP53 P04637 2/20 0.49
CYP3A4 P08684 1/20 0.48
MAPT P10636 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6448599 0.86 ALDH1A1 (0.67) ALDH1A1TACR3HPGDPTGFRLMNA
SCHEMBL5945348 0.81 DHODH (0.63) ALDH1A1TACR3PTGFRMAPTSMN1; SMN2
SCHEMBL5945399 0.81 PDE10A (0.68) TACR3
Hydrochloric Acid SCHEMBL6848801 0.80 DHODH (0.61) ALDH1A1TACR3PTGFRMAPTSMN1; SMN2
SCHEMBL4471465 0.80 TACR3 (0.82) ALDH1A1TACR3TP53CYP3A4SMN1; SMN2
SCHEMBL4471472 0.80 TACR3 (0.82) ALDH1A1TACR3TP53CYP3A4SMN1; SMN2
SCHEMBL4459968 0.79 DHODH (0.57) ALDH1A1TACR3PTGFRMAPTSMN1; SMN2
SCHEMBL6448666 0.76 TACR3 (0.60) ALDH1A1TACR3HPGDLMNATP53
SCHEMBL6449830 0.76 TACR3 (0.61) ALDH1A1TACR3HPGDLMNATP53
SCHEMBL6451528 0.75 LMNA (0.66) ALDH1A1TACR3HPGDLMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1517708-A1 COMBINATION TREATMENT FOR DEPRESSION AND ANXIETY BY NK1 AND NK3 ANTAGONISTS Pfizer Products Inc. (US) 2005-03-30 EP claimed
WO-2004000355-A1 COMBINATION TREATMENT FOR DEPRESSION AND ANXIETY BY NK1 AND NK3 ANTAGONISTS PFIZER PRODUCTS INC. (US) 2003-12-31 WO claimed
EP-1517708-A1 COMBINATION TREATMENT FOR DEPRESSION AND ANXIETY BY NK1 AND NK3 ANTAGONISTS Pfizer Products Inc. (US) 2005-03-30 EP disclosed
WO-2004000355-A1 COMBINATION TREATMENT FOR DEPRESSION AND ANXIETY BY NK1 AND NK3 ANTAGONISTS PFIZER PRODUCTS INC. (US) 2003-12-31 WO disclosed