SCHEMBL646139

SCHEMBL646139

Cc1cn(N)c(=O)[nH]c1=O

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.59
MAPK1 P28482 1/20 0.47
HPGD P15428 1/20 0.46
CRBN Q96SW2 1/20 0.41
ALDH1A1 P00352 2/20 0.40
TYMP P19971 2/20 0.40
LMNA P02545 1/20 0.40
ALB P02768 1/20 0.40
POLB P06746 1/20 0.40
ADRA1A P35348 1/20 0.40
BLM P54132 1/20 0.40
TK1 P04183 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15422063 0.78
SCHEMBL16248 0.76 MAPK1 (0.47) MAPK1HPGDCRBNALDH1A1TYMP
SCHEMBL17041835 0.76 TDP1 (0.53) TDP1MAPK1HPGDCRBNPOLB
SCHEMBL400005 0.74 TDP1 (1.00) TDP1CRBNALDH1A1POLB
SCHEMBL9192075 0.74 TDP1 (0.57) TDP1HPGDCRBNALDH1A1TYMP
SCHEMBL5176789 0.74 MAPK1 (0.46) TDP1MAPK1HPGDALDH1A1TYMP
SCHEMBL710870 0.74 MAPK1 (0.46) MAPK1HPGDALDH1A1TYMPLMNA
SCHEMBL9190653 0.74 TDP1 (0.57) TDP1CRBNTYMPBLMTK1
SCHEMBL9192590 0.74 TDP1 (0.57) TDP1HPGDCRBNALDH1A1LMNA
SCHEMBL7141531 0.74 MAPK1 (0.46) MAPK1HPGDALDH1A1TYMPLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 44 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250059537-A1 THERAPEUTIC OLIGONUCLEOTIDES HAVING AN INTER-NUCLEOSIDE AMIDE LINKAGE OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2025-02-20 US disclosed
EP-4448541-A1 THERAPEUTIC OLIGONUCLEOTIDES HAVING AN INTER-NUCLEOSIDE AMIDE LINKAGE Oxford University Innovation Limited (GB) 2024-10-23 EP disclosed
WO-2023178230-A1 PHOSPHORODIAMIDATE MORPHOLINO OLIGOMER CONJUGATES SAREPTA THERAPEUTICS, INC. (US) 2023-09-21 WO disclosed
WO-2023111597-A1 THERAPEUTIC OLIGONUCLEOTIDES HAVING AN INTER-NUCLEOSIDE AMIDE LINKAGE OXFORD UNIVERSITY INNOVATION LIMITED (GB) 2023-06-22 WO disclosed
EP-4115908-A1 EXON SKIPPING OLIGOMER CONJUGATES FOR MUSCULAR DYSTROPHY Sarepta Therapeutics, Inc. (US) 2023-01-11 EP disclosed
WO-2021108640-A1 COMPOUNDS AND METHODS FOR THE TREATMENT OF DUCHENNE MUSCULAR DYSTROPHY DTX PHARMA, INC. (US) 2021-06-03 WO disclosed
WO-2021108662-A1 COMPOUND COMPRISING A NUCLEIC ACID AND A HALF-LIFE EXTENSION MOTIF DTX PHARMA, INC. (US) 2021-06-03 WO disclosed
WO-2021000380-A1 MODIFIED NUCLEOSIDE, NUCLEOTIDE AND MODIFIED NUCLEIC ACID POLYMER, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF 中国人民解放军军事科学院军事医学研究院 2021-01-07 WO disclosed
US-10871467-B2 Cannabinoid profiling using nanopore transduction Cannaptic Biosciences, LLC (US) 2020-12-22 US disclosed
US-10822607-B2 Site-specific induction of bimolecular quadruplex-duplex hybrids and methods of using the same NANYANG TECHNOLOGICAL UNIVERSITY (SG) 2020-11-03 US disclosed
WO-2001016365-A1 POLY(ETHER-THIOETHER), POLY(ETHER-SULFOXIDE) AND POLY(ETHER-SULFONE) NUCLEIC ACIDS BIO-RAD LABORATORIES, INC. (US) 2001-03-08 WO disclosed
CN-1236395-A Real-time homogeneous nucleotide assay EDWARD E WINGER (US) 1999-11-24 CN disclosed
US-5773571-A BOND TO RNA AND DNA STRANDS NIELSEN PETER E (DK) 1998-06-30 US disclosed
EP-0688364-A4 GENETICALLY ENGINEERED ENZYMES AND THEIR CONJUGATES FOR DIAGNOSTIC ASSAYS ABBOTT LAB (US) 1997-10-15 EP disclosed
US-5539082-A Peptide nucleic acids NIELSEN PETER E (DK) 1996-07-23 US disclosed
EP-0699208-A1 NOVEL PEPTIDE NUCLEIC ACIDS NIELSEN, Peter Eigil (DK) 1996-03-06 EP disclosed
EP-0688364-A1 GENETICALLY ENGINEERED ENZYMES AND THEIR CONJUGATES FOR DIAGNOSTIC ASSAYS ABBOTT LABORATORIES (US) 1995-12-27 EP disclosed
WO-1994020636-A9 GENETICALLY ENGINEERED ENZYMES AND THEIR CONJUGATES FOR DIAGNOSTIC ASSAYS 1994-11-24 WO disclosed
WO-1994025477-A2 NOVEL PEPTIDE NUCLEIC ACIDS NIELSEN PETER E (DK) 1994-11-10 WO disclosed
WO-1994020636-A1 GENETICALLY ENGINEERED ENZYMES AND THEIR CONJUGATES FOR DIAGNOSTIC ASSAYS ABBOTT LABORATORIES (US) 1994-09-15 WO disclosed