SCHEMBL6463837

SCHEMBL6463837

CCCCN(C(=O)O)C(=O)N(CCc1nc(C(=O)NC(c2ccccc2)c2ccccc2)co1)CCc1ccccc1O

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.35
HTR1A P08908 1/20 0.34
TLR8 Q9NR97 1/20 0.33
C3AR1 Q16581 2/20 0.33
TACR3 P29371 2/20 0.32
HPGDS O60760 1/20 0.32
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
LMNA P02545 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HTT P42858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17749482 0.64 HDAC1 (0.50) TACR3HPGDSALDH1A1HDAC1HDAC8
Bicarbonate SCHEMBL4267974 0.58 BID (0.58) HTR1AKDM4ETSHRHSD17B10
SCHEMBL6833434 0.58 CA12 (0.50) ALDH1A1LMNAHPGDTSHRHSD17B10
Acetic Acid SCHEMBL9815548 0.57 BID (0.57) HTR1AKDM4ETSHRHSD17B10
SCHEMBL9777892 0.57 HTR1A (0.75) HTR1ATSHRHTT
SCHEMBL10964245 0.57 HTR1A (0.75) HTR1ATSHRHTT
Benzene SCHEMBL9052791 0.56 HTR1A (0.58) HTR1ATSHRHTT
Bicarbonate SCHEMBL9175297 0.56 BID (0.69) KDM4ETSHRHSD17B10HTT
Bicarbonate SCHEMBL4863706 0.56 BID (0.69) KDM4ETSHRHSD17B10HTT
SCHEMBL16333188 0.56 HTR1A (0.54) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed