SCHEMBL6466254

SCHEMBL6466254

Oc1ccc(CCNCC[C@@H](O)c2ccc(O)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.56
ADRB1 P08588 4/20 0.51
LMNA P02545 3/20 0.51
HIF1A Q16665 3/20 0.51
SLC6A4 P31645 3/20 0.51
OPRM1 P35372 3/20 0.51
SLC6A3 Q01959 2/20 0.51
SLC6A2 P23975 2/20 0.51
OPRK1 P41145 2/20 0.51
CYP2D6 P10635 1/20 0.51
GALR3 O60755 1/20 0.51
ADRA1A P35348 1/20 0.51
ALDH1A1 P00352 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
SLC22A1 O15245 1/20 0.51
CHRM2 P08172 1/20 0.51
CYP3A4 P08684 1/20 0.51
CHRM1 P11229 1/20 0.51
TSHR P16473 1/20 0.51
NFKB1 P19838 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10571063 0.83 KCNH2 (0.60) OPRK1SIGMAR1KCNH2
SCHEMBL2964767 0.81 ADRB2 (0.62) ADRB2ADRB1LMNAHIF1ASLC6A4
SCHEMBL7381628 0.81 TMEM97 (0.67) ADRB2ADRB1SLC6A2OPRK1ALDH1A1
SCHEMBL11611111 0.78 KCNH2 (0.77) ADRB2OPRK1SIGMAR1KCNH2
SCHEMBL4467889 0.77 ADRB2 (0.73) ADRB2ADRB1LMNAHIF1ASLC6A4
SCHEMBL9543386 0.77 ADRB2 (0.73) ADRB2ADRB1LMNAHIF1ASLC6A4
SCHEMBL4467885 0.77 ADRB2 (0.73) ADRB2ADRB1LMNAHIF1ASLC6A4
SCHEMBL10912498 0.75 ADRB2 (0.61) ADRB2ADRB1LMNAHIF1ASLC6A4
SCHEMBL11468342 0.75 ADRB2 (0.59) ADRB2ADRB1LMNAHIF1ASLC6A4
SCHEMBL11468343 0.75 ADRB2 (0.59) ADRB2ADRB1LMNAHIF1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1597229-A2 PYRROLIDINE DERIVATIVES AS OXYTOCIN ANTAGONISTS Applied Research Systems ARS Holding N.V. (AN) 2005-11-23 EP disclosed
WO-2004076407-A2 PYRROLIDINE DERIVATIVES AS OXYTOCIN ANTAGONISTS APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (NL) 2004-09-10 WO disclosed