SCHEMBL6466743

SCHEMBL6466743

CCc1[nH]c(CC)c(-c2ccc(C#N)cc2)c1C#N

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.44
GRIA2 P42262 1/20 0.44
GRIA4 P48058 1/20 0.44
AR P10275 4/20 0.41
PDE9A O76083 3/20 0.39
PGR P06401 1/20 0.39
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP11B2 P19099 2/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
HPGD P15428 1/20 0.38
MAPT P10636 1/20 0.37
KIF11 P52732 1/20 0.37
FNTA P49354 2/20 0.36
FNTB P49356 2/20 0.36
MMP3 P08254 1/20 0.36
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4910488 0.87 AR (0.43) CYP2A6GRIA2GRIA4ARPDE9A
SCHEMBL4922378 0.87 AR (0.43) CYP2A6GRIA2GRIA4ARPDE9A
SCHEMBL6469338 0.77 GRIA2 (0.48) CYP2A6GRIA2GRIA4ARPGR
SCHEMBL6464882 0.76 MAP2 (0.43) CYP2A6GRIA2GRIA4ARPGR
SCHEMBL4918690 0.75 MEN1 (0.43) CYP2A6GRIA2GRIA4ARPDE9A
SCHEMBL6466109 0.74 ALDH1A1 (0.59) CYP2A6GRIA2GRIA4ARPGR
SCHEMBL14154969 0.73 KDM4E (0.42) PDE9ATSHRHSD17B10ALDH1A1GAA
SCHEMBL4910473 0.73 KMT2A (0.44) CYP2A6GRIA2GRIA4ARPDE9A
SCHEMBL14154918 0.73 KDM4E (0.42) PDE9ATSHRHSD17B10ALDH1A1GAA
SCHEMBL4919125 0.72 GRIA2 (0.46) GRIA2GRIA4ARHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050101657-A1 Pyrrole derivatives for preventing or treating cancer sensitive to hormones; administered with luteininzing hormone releasing hormone derivative TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 2005-05-12 US disclosed
EP-1466902-A1 ANDROGEN RECEPTOR ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2004-10-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050101657-A1 Pyrrole derivatives for preventing or treating cancer sensitive to hormones; administered with luteininzing hormone releasing hormone derivative SHBG, PRLHR, FSHR CYP2A6 915/4885GRIA2 715/4885GRIA4 665/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.