SCHEMBL6467441

SCHEMBL6467441

O=C(CCc1ccccc1C(F)(F)F)N[C@@H](CCc1ccccc1)C(O)c1nc2ccccc2o1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 4/20 0.45
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
FAAH O00519 1/20 0.39
CES1 P23141 1/20 0.39
DAGLA Q9Y4D2 1/20 0.39
PTPN2 P17706 3/20 0.38
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
CNR2 P34972 1/20 0.37
XDH P47989 1/20 0.36
EPHX2 P34913 2/20 0.36
NR3C2 P08235 1/20 0.35
RBP4 P02753 1/20 0.35
FFAR2 O15552 1/20 0.35
PTGFR P43088 1/20 0.35
P2RY14 Q15391 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6462287 0.88 FAAH (0.44) POLBGAAFAAHCES1DAGLA
SCHEMBL7042871 0.83 PTPN1 (0.43) PTPN1PTPN2EPHX2
SCHEMBL6463429 0.81 DAGLA (0.47) PTPN1POLBGAAFAAHCES1
SCHEMBL6466336 0.81 MEN1 (0.40) FAAHCES1DAGLAEPHX2
SCHEMBL6473321 0.80 MEN1 (0.40) FAAHCES1DAGLAEPHX2
SCHEMBL6463649 0.80 MEN1 (0.40) FAAHCES1DAGLAEPHX2
SCHEMBL6462563 0.79 KDM4E (0.43) PTPN1CNR2
SCHEMBL5731227 0.76 CTSK (0.46) XDHEPHX2
SCHEMBL5731226 0.76 CTSK (0.46) XDHEPHX2
Hydrochloric Acid SCHEMBL6466455 0.75 SMN1; SMN2 (0.36) POLBFAAHCES1DAGLAXDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed