SCHEMBL6463649

SCHEMBL6463649

O=C(CCC1CCCCC1)N[C@@H](CCc1ccccc1)C(O)c1nc2ccccc2o1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
RAB9A P51151 2/20 0.40
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
BMP1 P13497 4/20 0.38
SOAT1 P35610 1/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
CTSS P25774 1/20 0.38
ALDH1A1 P00352 3/20 0.38
EPHX2 P34913 1/20 0.38
HPGD P15428 3/20 0.37
TDP1 Q9NUW8 1/20 0.37
FAAH O00519 1/20 0.37
CES1 P23141 1/20 0.37
DAGLA Q9Y4D2 1/20 0.37
NPC1 O15118 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6473321 1.00 MEN1 (0.40) MEN1KMT2ARAB9ALMNAMAPT
SCHEMBL6466336 0.99 MEN1 (0.40) MEN1KMT2ARAB9ALMNAMAPT
SCHEMBL6465745 0.90 KMT2A (0.43) MEN1KMT2ARAB9ALMNACTSL
SCHEMBL6465251 0.90 LMNA (0.40) MEN1KMT2ARAB9ALMNAMAPT
SCHEMBL7186564 0.88 MMP1 (0.39) MEN1KMT2ARAB9ACTSLCTSB
SCHEMBL7042906 0.87 DAGLA (0.46) MEN1KMT2ARAB9ALMNAMAPT
SCHEMBL7047598 0.87 CTSL (0.40) KMT2ALMNAMAPTCTSLCTSS
SCHEMBL6462287 0.86 FAAH (0.44) RAB9ALMNAMAPTHPGDFAAH
SCHEMBL6466278 0.85 BMP1 (0.36) MEN1KMT2ARAB9ALMNAMAPT
SCHEMBL7047934 0.85 CTSS (0.46) CTSLCTSBCTSSMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed