SCHEMBL6468002

SCHEMBL6468002

COC(=O)c1cc2c(c(C(=O)O)c1)CCCO2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.42
ALDH1A1 P00352 5/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
TP53 P04637 2/20 0.42
GLA P06280 1/20 0.42
GAA P10253 1/20 0.42
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
HSD17B10 Q99714 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
SMN1; SMN2 Q16637 2/20 0.40
MAPT P10636 2/20 0.38
POLB P06746 1/20 0.38
CTNNB1 P35222 1/20 0.37
WNT3A P56704 1/20 0.37
MAPK1 P28482 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12284075 0.96 ALDH1A1 (0.41) KDM4EALDH1A1MEN1KMT2ATP53
SCHEMBL2559609 0.92 KDM4E (0.47) KDM4EALDH1A1MEN1KMT2ATP53
SCHEMBL10069355 0.92 KDM4E (0.44) KDM4EALDH1A1MEN1KMT2ATP53
SCHEMBL6468123 0.89 KDM4E (0.44) KDM4EALDH1A1MEN1KMT2ATP53
SCHEMBL2556818 0.87 KDM4E (0.46) KDM4EALDH1A1MEN1KMT2ATP53
SCHEMBL2558486 0.85 NPC1 (0.44) KDM4EALDH1A1MEN1KMT2ATP53
SCHEMBL10069323 0.82 KDM4E (0.49) KDM4EALDH1A1MEN1KMT2ATP53
SCHEMBL10069338 0.80 KDM4E (0.47) KDM4EALDH1A1MEN1KMT2ATP53
SCHEMBL10069342 0.80 NPC1 (0.39) KDM4EALDH1A1MEN1KMT2ATP53
SCHEMBL10069318 0.80 ALDH1A1 (0.39) KDM4EALDH1A1MEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102958912-B Benzohydrol derivatives, a preparation process and pharmaceutical use thereof SHANGHAI HENGRUI PHARM CO LTD 2015-01-14 CN disclosed
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed
CN-102372653-A Diphenyl methanol derivative, preparation method thereof and application of diphenyl methanol derivative in medicine JIANGSU HENGRUI MEDICINE CO 2012-03-14 CN disclosed
WO-2012019428-A1 BENZOHYDROL DERIVATIVES, A PREPARATION PROCESS AND PHARMACEUTICAL USE THEREOF 上海恒瑞医药有限公司 (CN) 2012-02-16 WO disclosed
WO-2011130383-A1 COMPOUNDS CONTAINING FUSED RINGS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2011-10-20 WO disclosed