SCHEMBL6468103

SCHEMBL6468103

COC(=O)c1cc(C(=O)O)cc(-c2ccccc2C#N)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSA P10619 1/20 0.41
ADORA2A P29274 5/20 0.41
ADORA1 P30542 2/20 0.41
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
CRHBP P24387 3/20 0.41
CRHR2 Q13324 3/20 0.41
HPGD P15428 2/20 0.41
KDM6B O15054 1/20 0.40
KDM5C P41229 1/20 0.40
KDM4C Q9H3R0 1/20 0.40
KDM2A Q9Y2K7 1/20 0.40
KDM3A Q9Y4C1 1/20 0.40
PRKDC P78527 1/20 0.40
ATM Q13315 1/20 0.40
ATR Q13535 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL2710667 0.93 PRKDC (0.39) CTSAADORA2AADORA1KDM4EALDH1A1
SCHEMBL2709818 0.86 ADORA2A (0.39) CTSAADORA2AADORA1KDM4EALDH1A1
SCHEMBL2710671 0.83 ADORA2A (0.37) CTSAADORA2AADORA1KDM4EALDH1A1
SCHEMBL6468264 0.82 MAPT (0.42) ADORA2AADORA1KDM4EALDH1A1HPGD
SCHEMBL2343635 0.77 TSHR (0.44) CTSAKDM4EALDH1A1CRHBPCRHR2
SCHEMBL3590080 0.73 GAA (0.60) SMN1; SMN2NPC1MAPTRAB9AGAA
SCHEMBL21144538 0.73 TSHR (0.61) KDM4EALDH1A1KDM6BKDM5CKDM4C
SCHEMBL23381741 0.72 HTT (0.49) ADORA2AKDM4EALDH1A1CRHBPCRHR2
SCHEMBL2070250 0.72 TGFBR1 (0.49) KDM4EALDH1A1CRHBPCRHR2PRKDC
SCHEMBL3596754 0.72 ACHE (0.64) KDM4EALDH1A1CRHBPCRHR2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed