SCHEMBL6468264

SCHEMBL6468264

CCCCOC(=O)c1cc(C(=O)OC)nc(-c2ccccc2C#N)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.42
ESR1 P03372 6/20 0.40
L3MBTL1 Q9Y468 3/20 0.40
MDH2 P40926 1/20 0.40
TSHR P16473 4/20 0.40
TDP1 Q9NUW8 2/20 0.40
CNR2 P34972 1/20 0.39
ADORA2A P29274 2/20 0.39
ADORA1 P30542 2/20 0.39
CYP1A2 P05177 5/20 0.38
CYP2C19 P33261 5/20 0.38
SMN1; SMN2 Q16637 4/20 0.38
LMNA P02545 3/20 0.38
MAPK1 P28482 2/20 0.38
CYP2D6 P10635 1/20 0.38
NR1H2 P55055 1/20 0.38
RNASEL Q05823 1/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP3A4 P08684 3/20 0.38
CYP2C9 P11712 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6468103 0.82 CTSA (0.41) MAPTTSHRTDP1ADORA2AADORA1
SCHEMBL2709818 0.81 ADORA2A (0.39) MAPTTDP1ADORA2AADORA1SMN1; SMN2
SCHEMBL2710671 0.78 ADORA2A (0.37) TDP1ADORA2AADORA1SMN1; SMN2ALDH1A1
SCHEMBL9277021 0.70 TSHR (0.71) ESR1L3MBTL1TSHRTDP1CYP1A2
SCHEMBL23250562 0.69 ESR1 (0.67) ESR1L3MBTL1TSHRTDP1CNR2
SCHEMBL28388797 0.69 ALDH1A1 (0.65) MAPTL3MBTL1TSHRTDP1SMN1; SMN2
SCHEMBL4525162 0.68 PDK2 (0.41) MAPTL3MBTL1TSHRTDP1CYP1A2
SCHEMBL14919190 0.67 L3MBTL1 (0.55) ESR1L3MBTL1TSHRTDP1CYP1A2
SCHEMBL2347995 0.67 ESR2 (0.46) L3MBTL1TSHRADORA2ASMN1; SMN2ALDH1A1
SCHEMBL6057190 0.67 HPGD (0.60) ESR1L3MBTL1TSHRTDP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012054510-A1 OXADIAZOLE COMPOUNDS WHICH INHIBIT BETA-SECRETASE ACTIVITY AND METHODS OF USE THEREOF COMENTIS, INC. (US) 2012-04-26 WO disclosed