SCHEMBL6468438

SCHEMBL6468438

CCCCN(C(=O)c1nc2ccccc2o1)C(=O)C(CS(=O)(=O)Cc1ccccc1)NC(=O)O

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
FAAH O00519 3/20 0.40
CES1 P23141 2/20 0.40
DAGLA Q9Y4D2 1/20 0.40
XDH P47989 2/20 0.38
HSF1 Q00613 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CTSS P25774 8/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
PTPN2 P17706 1/20 0.36
PTPN1 P18031 1/20 0.36
PPARG P37231 1/20 0.35
PPARD Q03181 1/20 0.35
PPARA Q07869 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6462866 0.93 FAAH (0.38) FAAHCES1DAGLAXDHHSF1
SCHEMBL6461829 0.88 CTSS (0.43) CTSSCYP3A4CYP2C9
SCHEMBL7045520 0.85 FAAH (0.36) FAAHCES1DAGLACTSSCYP3A4
SCHEMBL6463182 0.85 CTSS (0.43) FAAHCES1CTSSCYP3A4CYP2C9
SCHEMBL7046391 0.84 FAAH (0.37) FAAHCES1DAGLAXDHALDH1A1
SCHEMBL6468151 0.84 FAAH (0.36) FAAHCES1XDHHSF1CTSS
SCHEMBL7049518 0.83 DAGLA (0.46) FAAHCES1DAGLAXDHALDH1A1
SCHEMBL7043169 0.82 CTSS (0.44) CTSSCYP3A4CYP2C9
SCHEMBL7043202 0.81 P2RY14 (0.37) FAAHCES1XDHHSF1CYP3A4
SCHEMBL6466564 0.80 DAGLA (0.41) FAAHCES1DAGLAALDH1A1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed
US-6576630-B1 Alkanoyl substituted benzooxazoles or naphthooxazoles AXYS PHARMACEUTICALS, INC. 2003-06-10 US disclosed