SCHEMBL6468151

SCHEMBL6468151

CCCCCN(C(=O)c1nc2ccccc2o1)C(=O)C(CS(=O)(=O)Cc1ccccc1OC(F)F)NC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FAAH O00519 2/20 0.36
CES1 P23141 1/20 0.36
PPARG P37231 6/20 0.34
PPARA Q07869 5/20 0.34
PPARD Q03181 3/20 0.34
HSF1 Q00613 1/20 0.33
XDH P47989 1/20 0.33
CTSS P25774 6/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6465211 0.90 CTSS (0.34) FAAHCES1PPARGPPARAPPARD
SCHEMBL6063906 0.89 CTSS (0.35) FAAHCES1PPARGPPARAPPARD
SCHEMBL6467367 0.86 CTSS (0.35) FAAHCES1HSF1CTSSCYP3A4
SCHEMBL6468438 0.84 FAAH (0.40) FAAHCES1PPARGPPARAPPARD
SCHEMBL7043202 0.84 P2RY14 (0.37) FAAHCES1PPARGPPARAPPARD
SCHEMBL6466172 0.84 FAAH (0.36) FAAHCES1PPARGPPARAPPARD
SCHEMBL6464590 0.81 CTSS (0.35) CTSS
SCHEMBL6462866 0.79 FAAH (0.38) FAAHCES1PPARGPPARAPPARD
SCHEMBL6461878 0.78 CTSS (0.37) FAAHCES1HSF1CTSS
SCHEMBL6466966 0.78 CTSS (0.37) FAAHCES1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP claimed
US-20030232864-A1 Novel Compounds and compositions as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2003-12-18 US claimed
US-6576630-B1 Alkanoyl substituted benzooxazoles or naphthooxazoles AXYS PHARMACEUTICALS, INC. 2003-06-10 US claimed
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed
US-20030232864-A1 Novel Compounds and compositions as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2003-12-18 US disclosed
US-6576630-B1 Alkanoyl substituted benzooxazoles or naphthooxazoles AXYS PHARMACEUTICALS, INC. 2003-06-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030232864-A1 Novel Compounds and compositions as protease inhibitors SERPINB1, CTRL, CTSZ FAAH 479/4885CES1 272/4885PPARG 4143/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.