SCHEMBL6468576

SCHEMBL6468576

NC(=O)c1ccc(CCCc2ccccc2)cc1-c1ccccc1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 9/20 0.53
PLA2G10 O15496 8/20 0.53
SLCO1B1 Q9Y6L6 1/20 0.49
ADRA1D P25100 1/20 0.43
BTK Q06187 1/20 0.43
FAAH O00519 2/20 0.42
SIRT2 Q8IXJ6 1/20 0.42
BRD4 O60885 1/20 0.42
BCAT2 O15382 1/20 0.41
PLA2G1B P04054 1/20 0.41
PLA2G5 P39877 1/20 0.41
PLA2G2C Q5R387 1/20 0.41
PLA2G12B Q9BX93 1/20 0.41
PLA2G12A Q9BZM1 1/20 0.41
PLA2G2F Q9BZM2 1/20 0.41
PLA2G3 Q9NZ20 1/20 0.41
PLA2G2E Q9NZK7 1/20 0.41
PLA2G2D Q9UNK4 1/20 0.41
LMNA P02545 1/20 0.41
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12394323 0.76 MCL1 (0.50) LMNANPC1ALDH1A1TP53GLA
SCHEMBL3789578 0.76 BTK (0.51) BTKBRD4BCAT2PLA2G1BLMNA
SCHEMBL27621512 0.74 BTK (0.50) BTKBRD4BCAT2ALDH1A1CYP3A4
SCHEMBL12394303 0.73 MAOB (0.52) ALDH1A1MAPK1SMN1; SMN2HDAC8MAOB
SCHEMBL1250166 0.73 BCAT2 (0.61) BTKBRD4BCAT2NPC1ALDH1A1
SCHEMBL7071495 0.71 HDAC1 (0.50) NPC1ALDH1A1MAPK1RAB9ASMN1; SMN2
SCHEMBL6685340 0.70 BTK (0.46) BTKBRD4BCAT2NPC1ALDH1A1
SCHEMBL23646005 0.69 PLA2G2A (1.00) PLA2G2APLA2G10SLCO1B1PLA2G1BPLA2G5
SCHEMBL30411519 0.69 PLA2G2A (1.00) PLA2G2APLA2G10SLCO1B1PLA2G1BPLA2G5
SCHEMBL3376462 0.69 SIRT2 (0.50) ADRA1DSIRT2LMNANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551795-A1 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2005-07-13 EP disclosed
WO-2004035525-A1 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE INC. (CA) 2004-04-29 WO disclosed