SCHEMBL6685340

SCHEMBL6685340

C#Cc1ccc(C(N)=O)c(-c2ccccc2N)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 1/20 0.46
BRD4 O60885 2/20 0.44
PDK2 Q15119 1/20 0.42
BCAT2 O15382 1/20 0.41
GRK6 P43250 1/20 0.40
PARP1 P09874 1/20 0.40
ALDH1A1 P00352 3/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
IKBKB O14920 2/20 0.37
AURKA O14965 1/20 0.35
RPS6KB1 P23443 1/20 0.35
MAP2K2 P36507 1/20 0.35
MAP2K1 Q02750 1/20 0.35
KDM4E B2RXH2 2/20 0.35
GAA P10253 1/20 0.35
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
CSNK1A1 P48729 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3789578 0.79 BTK (0.51) BTKBRD4BCAT2GRK6ALDH1A1
SCHEMBL27621512 0.78 BTK (0.50) BTKBRD4PDK2BCAT2GRK6
SCHEMBL1250166 0.76 BCAT2 (0.61) BTKBRD4BCAT2GRK6ALDH1A1
SCHEMBL28021807 0.74 BCAT2 (0.59) PDK2BCAT2PARP1ALDH1A1IKBKB
SCHEMBL18163775 0.72 ALDH1A1 (0.45) PDK2PARP1ALDH1A1AURKARPS6KB1
SCHEMBL16684995 0.71 BTK (0.53) BTKBRD4PDK2BCAT2GRK6
SCHEMBL2745941 0.71 CYP1A2 (0.41) ALDH1A1KDM4EGAANPC1RAB9A
SCHEMBL3379668 0.70 KMT2A (0.49) PARP1ALDH1A1AURKARPS6KB1MAP2K2
SCHEMBL17529586 0.70 PARP1 (0.42) PDK2PARP1ALDH1A1AURKARPS6KB1
SCHEMBL6468576 0.70 PLA2G2A (0.53) BTKBRD4BCAT2ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1429765-A2 INHIBITORS OF HISTONE DEACETYLASE Methylgene, Inc. (CA) 2004-06-23 EP disclosed
WO-2003024448-A2 INHIBITORS OF HISTONE DEACETYLASE METHYLGENE, INC. (CA) 2003-03-27 WO disclosed