SCHEMBL6469296

SCHEMBL6469296

CS(=O)(=O)c1ccc(-c2[nH]nc(CCO[N+](=O)[O-])c2-c2ccccn2)cc1

nearest known ligand 0.50

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.42
PTGS2 P35354 5/20 0.42
PTGS1 P23219 1/20 0.40
TGFBR1 P36897 1/20 0.39
SCD O00767 1/20 0.39
PKM P14618 1/20 0.37
CBFB Q13951 1/20 0.36
GPR39 O43194 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6590005 0.80 PTGS2 (0.43) ESR2PTGS2PTGS1
SCHEMBL6470491 0.77 PTGS2 (0.41) ESR2PTGS2PTGS1
SCHEMBL6441194 0.76 PTGS2 (0.46) ESR2PTGS2PTGS1
SCHEMBL6438018 0.74 PTGS2 (0.43) ESR2PTGS2PTGS1
SCHEMBL3865463 0.73 ESR2 (0.49) ESR2PTGS2PTGS1
SCHEMBL6440855 0.71 PTGS2 (0.42) ESR2PTGS2PTGS1
SCHEMBL4958540 0.71 PTGS2 (0.44) ESR2PTGS2PTGS1
SCHEMBL6438240 0.71 PTGS2 (0.48) ESR2PTGS2PTGS1
SCHEMBL6441773 0.71 PTGS2 (0.40) ESR2PTGS2PTGS1
SCHEMBL5150520 0.71 ESR2 (0.47) ESR2PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed