SCHEMBL4958540

SCHEMBL4958540

CS(=O)(=O)c1ccc(-c2[nH]nc(CO[N+](=O)[O-])c2Cc2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.44
PTGS1 P23219 5/20 0.39
ESR2 Q92731 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6590005 0.89 PTGS2 (0.43) PTGS2PTGS1ESR2
SCHEMBL4959110 0.82 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL4957579 0.79 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL4958867 0.77 PTGS2 (0.46) PTGS2PTGS1
SCHEMBL6439880 0.74 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL6441194 0.74 PTGS2 (0.46) PTGS2PTGS1ESR2
SCHEMBL8487155 0.73 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL6469296 0.71 ESR2 (0.42) PTGS2PTGS1ESR2
SCHEMBL6438455 0.69 PTGS2 (0.43) PTGS2PTGS1
SCHEMBL6441112 0.69 GHSR (0.40) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1542972-A4 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-01-23 EP claimed
EP-1542972-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-22 EP claimed
WO-2004010945-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-02-05 WO claimed
EP-1542972-A4 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2008-01-23 EP disclosed
EP-1542972-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-22 EP disclosed
WO-2004010945-A2 CYCLOOXYGENASE- 2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-02-05 WO disclosed