SCHEMBL6470815

SCHEMBL6470815

[AsH2]CC(c1ccccc1)c1nnn[nH]1

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.34
TAAR1 Q96RJ0 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
KDM4E B2RXH2 1/20 0.34
HRH1 P35367 3/20 0.32
HPGD P15428 1/20 0.32
NISCH Q9Y2I1 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
KMT2A Q03164 1/20 0.32
ATM Q13315 1/20 0.32
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7819515 0.81 HTR2A (0.39) HTR2ATAAR1L3MBTL1KDM4EHRH1
SCHEMBL5642404 0.81 HTR2A (0.54) HTR2ATAAR1HRH1HPGDSLC6A2
SCHEMBL9531756 0.80 SLC6A2 (0.50) HTR2ATAAR1L3MBTL1KDM4EHRH1
SCHEMBL11531757 0.76 KMT2A (0.35) HTR2ATAAR1L3MBTL1KDM4ESLC6A2
SCHEMBL7510243 0.76 KMT2A (0.44) L3MBTL1KDM4ESLC6A2SLC6A4SLC6A3
SCHEMBL3813663 0.74 TBXAS1 (0.37) HTR2AHRH1
SCHEMBL7438313 0.74 SLC6A2 (0.40) HPGDNISCHSLC6A2SLC6A4SLC6A3
SCHEMBL11528941 0.73 CYP1A2 (0.42) TAAR1SLC6A2SLC6A4SLC6A3
SCHEMBL9384051 0.73 DPP4 (0.39) KMT2AATM
SCHEMBL8090152 0.73 KMT2A (0.33) L3MBTL1KDM4ESLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603890-A1 TETRAZOLE AND OXADIAZOLONE SUBSTITUTED &bgr;-AMINO ACID DERIVATIVES Warner-Lambert Company LLC (US) 2005-12-14 EP disclosed
WO-2004078734-A1 TETRAZOLE AND OXADIAZOLONE SUBSTITUTED β-AMINO ACID DERIVATIVES WARNER-LAMBERT COMPANY LLC (US) 2004-09-16 WO disclosed