SCHEMBL8090152

SCHEMBL8090152

BrC(c1ccccc1)c1nnn[nH]1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
TRPA1 O75762 1/20 0.33
ATM Q13315 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 2/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
SLC6A2 P23975 2/20 0.31
SLC6A4 P31645 2/20 0.31
SLC6A3 Q01959 2/20 0.31
CFTR P13569 1/20 0.31
GOPC Q9HD26 1/20 0.31
CYP19A1 P11511 1/20 0.31
GAA P10253 1/20 0.31
DPP4 P27487 2/20 0.30
F2 P00734 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9090435 0.80 CES2 (0.33) KMT2ACES2CES1ATML3MBTL1
SCHEMBL11531757 0.79 KMT2A (0.35) KMT2AATML3MBTL1KDM4EALDH1A1
SCHEMBL7510243 0.79 KMT2A (0.44) KMT2AATML3MBTL1KDM4EALDH1A1
SCHEMBL27543188 0.78 KMT2A (0.34) KMT2AATML3MBTL1KDM4EALDH1A1
SCHEMBL9090443 0.76 SMN1; SMN2 (0.46) L3MBTL1KDM4EALDH1A1
SCHEMBL9384051 0.76 DPP4 (0.39) KMT2AATMDPP4F2
SCHEMBL8090075 0.76 TSHR (0.39) KMT2AATML3MBTL1KDM4EALDH1A1
SCHEMBL7679328 0.76 KMT2A (0.41) KMT2AATMKDM4EALDH1A1
Hydrochloric Acid SCHEMBL9985742 0.74 DPP4 (0.38) KMT2AATMALDH1A1DPP4F2
SCHEMBL7819515 0.73 HTR2A (0.39) L3MBTL1KDM4ESLC6A2SLC6A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0829480-B1 Tetrazolyl-substituted quinuclidines as substance P antagonists PFIZER (US) 2000-12-20 EP disclosed
US-5939434-A Tetrazolyl-substituted quinuclidines as substance P antagonists PFIZER PHARMACEUTICALS INC. (JP) 1999-08-17 US disclosed
EP-0829480-A2 Tetrazolyl-substituted quinuclidines as substance P antagonists PFIZER INC. (US) 1998-03-18 EP disclosed