SCHEMBL6473296

SCHEMBL6473296

CCCCCCCCCCC(Oc1ccccc1[N+](=O)[O-])C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.55
HPGD P15428 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.53
KMT2A Q03164 2/20 0.49
CTRC Q99895 1/20 0.48
ALDH1A1 P00352 6/20 0.44
HTT P42858 1/20 0.44
MEN1 O00255 1/20 0.44
TDP1 Q9NUW8 1/20 0.43
PPARG P37231 3/20 0.43
PTGES O14684 1/20 0.43
ALOX5 P09917 1/20 0.43
RAB9A P51151 2/20 0.42
NPC1 O15118 1/20 0.42
RECQL P46063 1/20 0.42
PPARA Q07869 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 1/20 0.40
LMNA P02545 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6256322 0.95 GAA (0.52) GAAHPGDL3MBTL1KMT2ACTRC
SCHEMBL11177445 0.89 GAA (0.57) GAAHPGDL3MBTL1KMT2AALDH1A1
SCHEMBL7508888 0.85 ALDH1A1 (0.51) GAAHPGDL3MBTL1KMT2AALDH1A1
SCHEMBL30639267 0.85 CTRC (0.54) KMT2ACTRCALDH1A1MEN1PPARG
Hydrochloric Acid SCHEMBL31748053 0.85 L3MBTL1 (0.45) GAAHPGDL3MBTL1KMT2AALDH1A1
SCHEMBL7692797 0.82 HPGD (0.54) GAAHPGDL3MBTL1KMT2AALDH1A1
SCHEMBL28327561 0.82 GAA (0.54) GAAHPGDL3MBTL1KMT2AALDH1A1
SCHEMBL7692800 0.82 HPGD (0.54) GAAHPGDL3MBTL1KMT2AALDH1A1
SCHEMBL21253070 0.81 CTRC (0.48) KMT2ACTRCALDH1A1MEN1PPARG
Hydrochloric Acid SCHEMBL8958669 0.81 HPGD (0.53) GAAHPGDL3MBTL1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005017106-A2 LIBRARIES OF OPTIMIZED CYTOCHROME P450 ENZYMES AND THE OPTIMIZED P450 ENZYMES CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2005-02-24 WO disclosed
WO-2003008563-A9 IMPROVED CYTOCHROME P450 OXYGENASES CALIFORNIA INST OF TECHN (US) 2003-08-14 WO disclosed
WO-2003008563-A2 IMPROVED CYTOCHROME P450 OXYGENASES CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2003-01-30 WO disclosed