SCHEMBL6476973

SCHEMBL6476973

CCCOc1ccccc1C(=O)Nc1c(CCC)c(Cl)n(C)c1C(N)=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNLIP P16233 1/20 0.44
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
MAPT P10636 3/20 0.42
NR1I2 O75469 1/20 0.42
LMNA P02545 1/20 0.42
CHRM2 P08172 1/20 0.42
CYP3A4 P08684 1/20 0.42
ADRA2A P08913 1/20 0.42
OPRK1 P41145 1/20 0.42
HTR2B P41595 1/20 0.42
SLC6A3 Q01959 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HIF1A Q16665 1/20 0.42
BRD4 O60885 1/20 0.41
NR3C1 P04150 1/20 0.40
MRGPRX1 Q96LB2 1/20 0.40
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6487627 0.93 MAPT (0.46) MEN1KMT2AMAPTRAB9ATP53
SCHEMBL6476050 0.89 KMT2A (0.43) PNLIPMEN1KMT2AMAPTNR1I2
SCHEMBL6481905 0.88 MAPT (0.42) PNLIPMEN1KMT2AMAPTNR1I2
SCHEMBL6476169 0.88 MEN1 (0.42) PNLIPMEN1KMT2AMAPTNR1I2
SCHEMBL6475637 0.82 MAPT (0.49) MEN1KMT2AMAPTRAB9ATP53
SCHEMBL6486828 0.81 MAPT (0.46) MEN1KMT2AMAPTRAB9ATP53
SCHEMBL6486467 0.81 MAPT (0.48) MEN1KMT2AMAPTLMNARAB9A
SCHEMBL6477006 0.80 MAPT (0.44) PNLIPMEN1KMT2AMAPTNR1I2
SCHEMBL1669 0.79 TERT (0.64) PNLIPMEN1KMT2AMAPTNR1I2
SCHEMBL8055429 0.74 TERT (0.56) PNLIPMEN1KMT2AMAPTNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6962911-B2 Pyrrolopyrimidinone derivatives, process of preparation and use SK CHEMICALS CO., LTD. (KR) 2005-11-08 US disclosed
EP-1257553-B1 PYRROLOPYRIMIDINONE DERIVATIVES, PROCESS OF PREPARATION AND USE SK CHEMICALS CO LTD (KR) 2004-05-26 EP disclosed
US-20030171361-A1 Pyrrolopyrimidinone derivatives, process of preparation and use SK CHEMICALS CO., LTD. (KR) 2003-09-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030171361-A1 Pyrrolopyrimidinone derivatives, process of preparation and use CYP2C19, DHPS, SDHA PNLIP 2491/4885MEN1 2829/4885KMT2A 4373/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.