Salubrinal

Salubrinal

SCHEMBL6477833

O=C(C=Cc1ccccc1)NC(NC(=S)Nc1cccc2cccnc12)C(Cl)(Cl)Cl

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 12/20 1.00
KMT2A Q03164 12/20 1.00
MAPT P10636 8/20 1.00
HPGD P15428 2/20 1.00
ALDH1A1 P00352 7/20 0.66
LMNA P02545 9/20 0.64
NPSR1 Q6W5P4 6/20 0.64
SMN1; SMN2 Q16637 5/20 0.61
HTT P42858 4/20 0.61
CYP1A2 P05177 2/20 0.59
CYP3A4 P08684 2/20 0.59
CYP2D6 P10635 2/20 0.59
CYP2C9 P11712 2/20 0.59
CYP2C19 P33261 2/20 0.59
ALOX12 P18054 1/20 0.59
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
KDM4E B2RXH2 2/20 0.49
RECQL P46063 2/20 0.49
MMP14 P50281 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Salubrinal SCHEMBL6477826 1.00 MEN1 (1.00) MEN1KMT2AMAPTHPGDALDH1A1
Salubrinal SCHEMBL17360638 1.00 MEN1 (1.00) MEN1KMT2AMAPTHPGDALDH1A1
SCHEMBL14782069 0.91 MEN1 (0.84) MEN1KMT2AMAPTHPGDALDH1A1
SCHEMBL21237547 0.89 MEN1 (0.81) MEN1KMT2AMAPTHPGDALDH1A1
SCHEMBL14819076 0.88 MEN1 (0.78) MEN1KMT2AMAPTHPGDALDH1A1
SCHEMBL16283211 0.88 KMT2A (0.78) MEN1KMT2AMAPTHPGDALDH1A1
SCHEMBL14819072 0.86 MEN1 (0.75) MEN1KMT2AMAPTHPGDALDH1A1
SCHEMBL17508602 0.86 MEN1 (0.75) MEN1KMT2AMAPTHPGDALDH1A1
SCHEMBL20438010 0.83 MEN1 (0.72) MEN1KMT2AMAPTHPGDALDH1A1
SCHEMBL28574843 0.81 MEN1 (0.68) MEN1KMT2AMAPTHPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118161473-A ISRIB application in preparing medicine for preventing and treating ischemic cerebral apoplexy 苏州大学 2024-06-11 CN claimed
EP-3820471-A1 TREATMENT OF CHRONIC TRAUMATIC ENCEPHALOPATHY CTEC LLC (US) 2021-05-19 EP claimed
US-6946474-B2 Nitrogen-containing compounds and their use as glycine transport inhibitors MERCK & CO., INC. (US) 2005-09-20 US claimed
JP-2004518628-A 2004-06-24 JP claimed
US-20040034069-A1 Nitrogen-containing compounds and their use as glycine transport inhibitors MERCK SHARP & DOHME CORP. 2004-02-19 US claimed
EP-1324986-A1 NITROGEN-CONTAINING COMPOUNDS AND THEIR USE AS GLYCINE TRANSPORT INHIBITORS GLIATECH, INC. (US) 2003-07-09 EP claimed
US-20020082283-A1 Nitrogen-containing compounds and their use as glycine transport inhibitors GLIATECH, INC. 2002-06-27 US claimed
WO-2002022581-A1 NITROGEN-CONTAINING COMPOUNDS AND THEIR USE AS GLYCINE TRANSPORT INHIBITORS GLIATECH, INC. (US) 2002-03-21 WO claimed
US-12157728-B2 Targeting of endoplasmic reticulum dysfunction and protein folding stress to treat neurological conditions ALS THERAPY DEVELOPMENT INSTITUTE (US) 2024-12-03 US disclosed
CN-118161473-A ISRIB application in preparing medicine for preventing and treating ischemic cerebral apoplexy 苏州大学 2024-06-11 CN disclosed
US-20230382890-A1 TARGETING OF ENDOPLASMIC RETICULUM DYSFUNCTION AND PROTEIN FOLDING STRESS TO TREAT NEUROLOGICAL CONDITIONS ALS THERAPY DEVELOPMENT INSTITUTE 2023-11-30 US disclosed
US-11708349-B2 Targeting of endoplasmic reticulum dysfunction and protein folding stress to treat neurological conditions ALS THERAPY DEVELOPMENT INSTITUTE (US) 2023-07-25 US disclosed
CN-116397028-A Application of copper death-related lncRNAs in lung squamous cell carcinoma prognosis evaluation 桂林医学院 2023-07-07 CN disclosed
EP-3820471-A1 TREATMENT OF CHRONIC TRAUMATIC ENCEPHALOPATHY CTEC LLC (US) 2021-05-19 EP disclosed
WO-2012140208-A1 SCREENING METHODS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF INFLAMMATORY BOWEL DISEASES INSERM (INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE) (FR) 2012-10-18 WO disclosed
US-6946474-B2 Nitrogen-containing compounds and their use as glycine transport inhibitors MERCK & CO., INC. (US) 2005-09-20 US disclosed
US-20040034069-A1 Nitrogen-containing compounds and their use as glycine transport inhibitors MERCK SHARP & DOHME CORP. 2004-02-19 US disclosed
EP-1324986-A1 NITROGEN-CONTAINING COMPOUNDS AND THEIR USE AS GLYCINE TRANSPORT INHIBITORS GLIATECH, INC. (US) 2003-07-09 EP disclosed
US-20020082283-A1 Nitrogen-containing compounds and their use as glycine transport inhibitors GLIATECH, INC. 2002-06-27 US disclosed
WO-2002022581-A1 NITROGEN-CONTAINING COMPOUNDS AND THEIR USE AS GLYCINE TRANSPORT INHIBITORS GLIATECH, INC. (US) 2002-03-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020082283-A1 Nitrogen-containing compounds and their use as glycine transport inhibitors SLC1A5, SLC6A7, SLC6A15 MEN1 1992/4885KMT2A 4212/4885MAPT 1381/4885
US-20230382890-A1 TARGETING OF ENDOPLASMIC RETICULUM DYSFUNCTION AND PROTEIN FOLDING STRESS TO TREAT NEUROLOGICAL CONDITIONS HSPA5, HSP90B1, HSPD1 MEN1 4712/4885KMT2A 4807/4885MAPT 10/4885
US-11708349-B2 Targeting of endoplasmic reticulum dysfunction and protein folding stress to treat neurological conditions HSPA5, HSP90B1, HSPD1 MEN1 4712/4885KMT2A 4807/4885MAPT 10/4885
US-20040034069-A1 Nitrogen-containing compounds and their use as glycine transport inhibitors SLC1A5, SLC6A7, SLC6A15 MEN1 1992/4885KMT2A 4212/4885MAPT 1381/4885
US-12157728-B2 Targeting of endoplasmic reticulum dysfunction and protein folding stress to treat neurological conditions HSPA5, HSP90B1, HSPD1 MEN1 4712/4885KMT2A 4807/4885MAPT 10/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.