SCHEMBL6478317

SCHEMBL6478317

COc1ccccc1CS(=O)(=O)C(CCCC(=O)c1nc2ccccc2o1)C(NC(=O)N(C)C)C(N)=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 3/20 0.38
CES1 P23141 2/20 0.38
DAGLA Q9Y4D2 1/20 0.38
P2RY14 Q15391 1/20 0.37
XDH P47989 2/20 0.37
NLRP3 Q96P20 2/20 0.37
TLR4 O00206 1/20 0.37
MAPT P10636 2/20 0.35
LMNA P02545 2/20 0.35
POLB P06746 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
RAB9A P51151 2/20 0.34
PSMD14 O00487 1/20 0.34
NPC1 O15118 1/20 0.34
TSHR P16473 2/20 0.34
HSD17B10 Q99714 2/20 0.34
USP2 O75604 1/20 0.34
ALOX12 P18054 1/20 0.34
CTSS P25774 5/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6463821 0.87 DAGLA (0.40) FAAHCES1DAGLAP2RY14XDH
SCHEMBL7045310 0.79 FAAH (0.38) FAAHCES1DAGLAP2RY14XDH
SCHEMBL6467434 0.78 HDAC6 (0.40) FAAHCES1DAGLAP2RY14XDH
SCHEMBL7047033 0.75 FAAH (0.41) FAAHCES1DAGLAP2RY14XDH
SCHEMBL6463510 0.75 FAAH (0.41) FAAHCES1DAGLAP2RY14XDH
SCHEMBL7043208 0.72 FAAH (0.41) FAAHCES1DAGLAP2RY14XDH
SCHEMBL6462832 0.72 DAGLA (0.43) FAAHCES1DAGLAP2RY14XDH
SCHEMBL6478314 0.72 CTSS (0.42) CTSS
SCHEMBL7188004 0.72 FAAH (0.39) FAAHCES1DAGLAXDHNLRP3
SCHEMBL7045307 0.72 CTSS (0.42) CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1516877-A1 Amine derivatives as protease inhibitors AXYS PHARMACEUTICALS, INC. (US) 2005-03-23 EP disclosed