SCHEMBL647941

SCHEMBL647941

O=C(O)OC(c1ccccc1)c1nccn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.38
KDM4E B2RXH2 1/20 0.38
KIF11 P52732 1/20 0.34
NCOA3 Q9Y6Q9 1/20 0.34
POLB P06746 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
LMNA P02545 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
HTR1A P08908 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
MAPT P10636 1/20 0.30
CYP19A1 P11511 3/20 0.30
CYP1A1 P04798 1/20 0.30
MEN1 O00255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20768154 0.75 KMT2A (0.38) KMT2AKDM4EPOLBCYP11B1CYP11B2
SCHEMBL9238656 0.73 KDM4E (0.44) KMT2AKDM4ECYP11B1CYP11B2MEN1
SCHEMBL27476843 0.69 CYP11B1 (0.40) KMT2AKDM4EESR1CYP11B1CYP11B2
SCHEMBL871451 0.69 ESR1 (0.57) KMT2AKDM4EKIF11ESR1ESR2
Hydrochloric Acid SCHEMBL11846585 0.67 ESR1 (0.55) KMT2AKDM4EKIF11ESR1ESR2
SCHEMBL4543871 0.67 CYP11B1 (0.43) KMT2ACYP11B1CYP11B2LMNAADRA1D
SCHEMBL1564248 0.67 KCNN4 (0.40) KMT2AKDM4EPOLBCYP11B1CYP11B2
SCHEMBL27469711 0.67 KMT2A (0.38) KMT2AKDM4EESR1CYP11B1CYP11B2
SCHEMBL6446028 0.66 KMT2A (0.43) KMT2AKDM4EESR1CYP11B1CYP11B2
SCHEMBL7246865 0.66 KDM4E (0.39) KDM4ECYP11B1CYP11B2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119665-B2 Aryl imidazoles and related compounds as C5a receptor modulators NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2012-02-21 US disclosed
US-8119687-B2 Derivatives of dioxan-2-alkyl carbamates, preparation thereof and application thereof in therapeutics SANOFI-AVENTIS (FR) 2012-02-21 US disclosed