SCHEMBL6482895

SCHEMBL6482895

O=C(CCc1cccnc1)NCCCCCCN1CCN(C2c3ccccc3CCc3ccccc32)CC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FNTA P49354 3/20 0.47
FNTB P49356 3/20 0.47
OPRL1 P41146 2/20 0.46
DRD3 P35462 3/20 0.44
DRD2 P14416 2/20 0.44
PTAFR P25105 2/20 0.44
HTR1A P08908 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HTR2A P28223 1/20 0.44
P2RX7 Q99572 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HTR7 P34969 1/20 0.42
C3AR1 Q16581 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3077208 0.99 FNTA (0.47) FNTAFNTBOPRL1DRD3DRD2
SCHEMBL6163043 0.89 ALDH1A1 (0.43) FNTAFNTBOPRL1DRD3DRD2
SCHEMBL6271049 0.86 OPRL1 (0.46) OPRL1DRD3DRD2PTAFRHTR1A
SCHEMBL3074401 0.80 DRD3 (0.57) OPRL1DRD3DRD2CYP3A4CYP2C9
SCHEMBL3074404 0.80 DRD3 (0.57) OPRL1DRD3DRD2CYP3A4CYP2C9
SCHEMBL3073089 0.80 DRD3 (0.57) OPRL1DRD3DRD2CYP3A4CYP2C9
SCHEMBL3073087 0.80 DRD3 (0.57) OPRL1DRD3DRD2CYP3A4CYP2C9
SCHEMBL7672874 0.80 CHRNA7 (0.57) DRD3DRD2PTAFRHTR1AALDH1A1
SCHEMBL21245369 0.80 HDAC8 (0.52) PTAFRALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL3081179 0.79 DRD2 (0.58) FNTAFNTBOPRL1DRD3DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6903118-B1 Piperazinyl-substituted pyridylalkane, alkene and alkine carboxamides KLINGE PHARMA GMBH (DE) 2005-06-07 US claimed