SCHEMBL6163043

SCHEMBL6163043

O=C(CCc1cccnc1)NCCCCN1CCN(C2c3ccccc3COc3ccccc32)CC1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
TBXAS1 P24557 2/20 0.42
DRD3 P35462 3/20 0.41
DRD2 P14416 2/20 0.41
ACHE P22303 1/20 0.41
OPRL1 P41146 1/20 0.41
PTAFR P25105 2/20 0.41
HTR1A P08908 1/20 0.41
HTR2A P28223 1/20 0.41
FNTA P49354 1/20 0.40
FNTB P49356 1/20 0.40
LMNA P02545 1/20 0.40
GAA P10253 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
RECQL P46063 1/20 0.40
C3AR1 Q16581 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3077208 0.90 FNTA (0.47) ALDH1A1DRD3DRD2OPRL1PTAFR
SCHEMBL6482895 0.89 FNTA (0.47) ALDH1A1DRD3DRD2OPRL1PTAFR
SCHEMBL3088918 0.89 LMNA (0.46) ALDH1A1TBXAS1ACHEPTAFRLMNA
SCHEMBL6268837 0.86 ACHE (0.46) ALDH1A1TBXAS1DRD3DRD2ACHE
SCHEMBL6777801 0.81 LMNA (0.43) ALDH1A1TBXAS1ACHEPTAFRLMNA
SCHEMBL6271049 0.77 OPRL1 (0.46) ALDH1A1DRD3DRD2OPRL1PTAFR
SCHEMBL7672874 0.77 CHRNA7 (0.57) ALDH1A1DRD3DRD2PTAFRHTR1A
SCHEMBL3458409 0.75 ALDH1A1 (0.63) ALDH1A1DRD3DRD2PTAFRHTR1A
SCHEMBL87991 0.74 LMNA (0.49) ALDH1A1PTAFRLMNACYP1A2CYP3A4
SCHEMBL3074297 0.74 TBXAS1 (0.35) TBXAS1DRD3HTR1AHTR2AFNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060163-B1 NEW PIPERAZINYL-SUBSTITUTED PYRIDYLALKANE, ALKENE AND ALKINE CARBOXAMIDES KLINGE CO CHEM PHARM FAB (DE) 2005-10-12 EP claimed