SCHEMBL6484201

SCHEMBL6484201

COc1ccccc1N1CCN(C(=O)CC(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.68
LMNA P02545 2/20 0.68
TSHR P16473 3/20 0.65
RAB9A P51151 1/20 0.65
L3MBTL1 Q9Y468 2/20 0.60
KDM4E B2RXH2 1/20 0.60
TDP1 Q9NUW8 1/20 0.60
CACNA2D1 P54289 3/20 0.60
CACNA1B Q00975 3/20 0.60
CACNB1 Q02641 3/20 0.60
CACNA1C Q13936 3/20 0.60
MEN1 O00255 1/20 0.59
MAPT P10636 1/20 0.59
HTT P42858 1/20 0.59
KMT2A Q03164 1/20 0.59
POLB P06746 1/20 0.59
SMN1; SMN2 Q16637 1/20 0.59
HTR7 P34969 1/20 0.58
CACNA1G O43497 1/20 0.58
ADRA1A P35348 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976802 0.93 CACNA2D1 (0.66) ALDH1A1LMNATSHRRAB9AL3MBTL1
Hydrochloric Acid SCHEMBL6482751 0.92 CACNA2D1 (0.65) ALDH1A1LMNATSHRRAB9AL3MBTL1
SCHEMBL6484058 0.88 HTR1A (0.63) ALDH1A1LMNATSHRRAB9AL3MBTL1
SCHEMBL6546626 0.83 ALDH1A1 (0.65) ALDH1A1LMNATSHRRAB9AKDM4E
SCHEMBL12781882 0.82 TSHR (0.73) ALDH1A1LMNATSHRRAB9AL3MBTL1
SCHEMBL20419343 0.82 TSHR (0.68) ALDH1A1LMNATSHRRAB9AL3MBTL1
SCHEMBL10586177 0.81 TSHR (0.71) ALDH1A1LMNATSHRRAB9AL3MBTL1
SCHEMBL13979787 0.81 TSHR (0.71) ALDH1A1LMNATSHRRAB9AL3MBTL1
SCHEMBL14500742 0.81 TSHR (0.71) ALDH1A1LMNATSHRRAB9AL3MBTL1
SCHEMBL8422424 0.81 ALDH1A1 (1.00) ALDH1A1LMNATSHRRAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6894052-B1 Serotonergic receptor antagonist RECORDATI S.A. CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 2005-05-17 US disclosed
EP-1000046-B1 PIPERAZINE DERIVATIVES ACTIVE ON THE LOWER URINARY TRACT RECORDATI CHEM PHARM (CH) 2003-11-26 EP disclosed
EP-1000046-A1 PIPERAZINE DERIVATIVES ACTIVE ON THE LOWER URINARY TRACT RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 2000-05-17 EP disclosed
WO-1999006383-A1 PIPERAZINE DERIVATIVES ACTIVE ON THE LOWER URINARY TRACT RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1999-02-11 WO disclosed