SCHEMBL6484692

SCHEMBL6484692

COc1ccccc1N1CCN(CCC(c2ccc([N+](=O)[O-])cc2)c2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.81
ADRA1D P25100 2/20 0.60
ADRA1A P35348 2/20 0.60
ADRA1B P35368 2/20 0.60
LMNA P02545 2/20 0.57
ALDH1A1 P00352 1/20 0.57
MAPT P10636 1/20 0.57
MAPK1 P28482 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.57
CCR2 P41597 1/20 0.55
MEN1 O00255 1/20 0.55
NPC1 O15118 1/20 0.55
CASP3 P42574 1/20 0.55
RAB9A P51151 1/20 0.55
KMT2A Q03164 1/20 0.55
SENP7 Q9BQF6 1/20 0.55
SENP6 Q9GZR1 1/20 0.55
DRD2 P14416 2/20 0.55
DRD3 P35462 1/20 0.55
HTR1D P28221 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6971387 0.99 HTR1A (0.79) HTR1AADRA1DADRA1AADRA1BLMNA
SCHEMBL6486972 0.86 HTR1A (0.79) HTR1AADRA1DADRA1AADRA1BDRD2
Hydrochloric Acid SCHEMBL6482862 0.85 HTR1A (0.77) HTR1AADRA1DADRA1AADRA1BDRD2
SCHEMBL6484702 0.84 HTR1A (0.78) HTR1AADRA1DADRA1AADRA1BALDH1A1
SCHEMBL6936851 0.83 HTR1A (0.69) HTR1AADRA1DADRA1AADRA1BLMNA
Hydrochloric Acid SCHEMBL6473994 0.83 HTR1A (0.77) HTR1AADRA1DADRA1AADRA1BALDH1A1
SCHEMBL6484058 0.81 HTR1A (0.63) HTR1ALMNAALDH1A1MAPTMAPK1
SCHEMBL11556531 0.81 MAPK1 (0.69) HTR1AADRA1DADRA1AADRA1BLMNA
SCHEMBL6936848 0.80 HTR1A (0.67) HTR1AADRA1DADRA1AADRA1BLMNA
SCHEMBL11860558 0.79 HTR1A (0.64) HTR1AADRA1DADRA1AADRA1BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6894052-B1 Serotonergic receptor antagonist RECORDATI S.A. CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 2005-05-17 US claimed
EP-1000046-B1 PIPERAZINE DERIVATIVES ACTIVE ON THE LOWER URINARY TRACT RECORDATI CHEM PHARM (CH) 2003-11-26 EP claimed
JP-2001512111-A 2001-08-21 JP claimed
EP-1000046-A1 PIPERAZINE DERIVATIVES ACTIVE ON THE LOWER URINARY TRACT RECORDATI S.A. CHEMICAL and PHARMACEUTICAL COMPANY (CH) 2000-05-17 EP claimed
WO-1999006383-A1 PIPERAZINE DERIVATIVES ACTIVE ON THE LOWER URINARY TRACT RECORDATI S.A., CHEMICAL AND PHARMACEUTICAL COMPANY (CH) 1999-02-11 WO claimed