SCHEMBL6489564

SCHEMBL6489564

CNCCC(Oc1cc(Cl)c(F)cc1C#N)c1cccnc1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 17/20 0.59
NOS2 P35228 13/20 0.59
SLC6A2 P23975 13/20 0.59
CYP2D6 P10635 11/20 0.59
KCNH2 Q12809 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL6491974 0.95 SLC6A4 (0.64) SLC6A4NOS2SLC6A2CYP2D6KCNH2
SCHEMBL6500286 0.88 NOS2 (0.76) SLC6A4NOS2SLC6A2CYP2D6KCNH2
SCHEMBL6490961 0.88 SLC6A4 (0.76) SLC6A4NOS2SLC6A2CYP2D6KCNH2
Oxalic Acid SCHEMBL6502548 0.83 SLC6A4 (0.78) SLC6A4NOS2SLC6A2CYP2D6KCNH2
Oxalic Acid SCHEMBL6502777 0.83 NOS2 (0.80) SLC6A4NOS2SLC6A2CYP2D6KCNH2
SCHEMBL6491537 0.83 SLC6A4 (0.53) SLC6A4NOS2SLC6A2CYP2D6KCNH2
Hydrochloric Acid SCHEMBL6490386 0.82 SLC6A4 (0.53) SLC6A4NOS2SLC6A2CYP2D6KCNH2
SCHEMBL6577152 0.81 NOS2 (0.67) SLC6A4NOS2SLC6A2CYP2D6KCNH2
SCHEMBL6497932 0.80 SLC6A4 (0.55) SLC6A4NOS2SLC6A2CYP2D6KCNH2
SCHEMBL6748032 0.80 NOS2 (0.55) SLC6A4NOS2SLC6A2CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1235870-C Novel use of phenyl hetero alkylamine derivatives ASTRAZENECA AB (SE) 2006-01-11 CN claimed
US-6887871-B2 Use of phenylheteroakylamine derivatives ASTRAZENECA AB (SE) 2005-05-03 US claimed
EP-1263711-B1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2004-12-15 EP claimed
US-20030158185-A1 Novel use of phenylheteroakylamine derivatives ASTRAZENECA AB (SE) 2003-08-21 US claimed
CN-1411435-A Novel use of phenylheteroalkylamine derivatives ASTRAZENECA AB (SE) 2003-04-16 CN claimed
CN-1235870-C Novel use of phenyl hetero alkylamine derivatives ASTRAZENECA AB (SE) 2006-01-11 CN disclosed
US-6887871-B2 Use of phenylheteroakylamine derivatives ASTRAZENECA AB (SE) 2005-05-03 US disclosed
EP-1263711-B1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2004-12-15 EP disclosed
US-20030158185-A1 Novel use of phenylheteroakylamine derivatives ASTRAZENECA AB (SE) 2003-08-21 US disclosed
CN-1411435-A Novel use of phenylheteroalkylamine derivatives ASTRAZENECA AB (SE) 2003-04-16 CN disclosed
EP-1263711-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES AstraZeneca AB (SE) 2002-12-11 EP disclosed
WO-2001062704-A1 NOVEL USE OF PHENYLHETEROALKYLAMINE DERIVATIVES ASTRAZENECA AB (SE) 2001-08-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030158185-A1 Novel use of phenylheteroakylamine derivatives NOS1, XDH, NOS2 SLC6A4 2468/4885NOS2 3/4885SLC6A2 1776/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.