SCHEMBL6489587

SCHEMBL6489587

N[C@@H]1CN2C(=O)N(c3cc(Cl)cc(Cl)c3)C(=O)[C@@]2(Cc2ccc(OC(F)(F)F)cc2)C1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
METAP2 P50579 1/20 0.37
HCRTR1 O43613 6/20 0.36
HCRTR2 O43614 6/20 0.36
ITGB2 P05107 1/20 0.36
ICAM1 P05362 1/20 0.36
ITGAL P20701 1/20 0.36
SCN9A Q15858 1/20 0.35
GRIN2B Q13224 1/20 0.35
CYP3A4 P08684 1/20 0.35
GRM2 Q14416 1/20 0.35
PRCP P42785 2/20 0.35
LIPE Q05469 5/20 0.34
AADAT Q8N5Z0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4847817 0.92 KCNN3 (0.38) METAP2HCRTR1HCRTR2CYP3A4GRM2
SCHEMBL14254856 0.89 METAP2 (0.39) METAP2HCRTR1HCRTR2ITGB2ICAM1
SCHEMBL4841746 0.89 METAP2 (0.39) METAP2HCRTR1HCRTR2ITGB2ICAM1
SCHEMBL4841580 0.87 METAP2 (0.39) METAP2HCRTR1HCRTR2ITGB2ICAM1
SCHEMBL4847332 0.84 ITGAL (0.52) ITGB2ICAM1ITGAL
SCHEMBL6478278 0.84 ITGAL (0.52) ITGB2ICAM1ITGAL
SCHEMBL4844861 0.83 METAP2 (0.39) METAP2HCRTR1HCRTR2SCN9ALIPE
SCHEMBL4848499 0.83 SCN9A (0.42) METAP2HCRTR1HCRTR2ITGB2ICAM1
SCHEMBL4848356 0.83 METAP2 (0.37) METAP2HCRTR1HCRTR2ITGB2ICAM1
SCHEMBL6490093 0.82 METAP2 (0.37) METAP2HCRTR1HCRTR2ITGB2ICAM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6897225-B1 Inhibitors of αLβ2 mediated cell adhesion TANABE SEIYAKU CO., LTD. (JP) 2005-05-24 US disclosed