SCHEMBL6489941

SCHEMBL6489941

CC(C)c1ccc2[nH]c3c(c2c1)C(=NNCC1=NCCN1)CC(c1ccccc1)C3

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 5/20 0.36
MAOA P21397 4/20 0.36
MAOB P27338 4/20 0.36
HTR1D P28221 2/20 0.35
HTR1B P28222 2/20 0.35
ADRA1D P25100 5/20 0.34
ADRA1A P35348 5/20 0.34
ADRA1B P35368 5/20 0.34
ADRA2A P08913 3/20 0.34
PIM1 P11309 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
ADRA2B P18089 3/20 0.32
ADRA2C P18825 3/20 0.32
LMNA P02545 2/20 0.32
HPGD P15428 2/20 0.32
HSD17B10 Q99714 2/20 0.32
KMT2A Q03164 1/20 0.32
ALDH1A1 P00352 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6489545 0.90 KMT2A (0.40) NISCHMAOAMAOBADRA1DADRA1A
SCHEMBL6500360 0.88 MAOA (0.37) NISCHMAOAMAOBADRA1DADRA1A
SCHEMBL6486887 0.81 MAPT (0.41) NISCHMAOAMAOBHTR1DHTR1B
SCHEMBL6489930 0.80 HPGD (0.33) ADRA2APIM1CLK4ADRA2BADRA2C
SCHEMBL6487105 0.80 HTR1D (0.38) NISCHMAOAMAOBHTR1DHTR1B
SCHEMBL6495347 0.76 MAPT (0.35) PIM1CLK4LMNAHPGDHSD17B10
SCHEMBL7128314 0.76 MAPT (0.35) PIM1CLK4LMNAHPGDHSD17B10
SCHEMBL6491133 0.70 ADRA2C (0.42) NISCHMAOAMAOBADRA1DADRA1A
SCHEMBL6488762 0.69 ADRA2C (0.40) NISCHMAOAMAOBADRA1DADRA1A
SCHEMBL6489539 0.69 ALDH1A1 (0.40) PIM1CLK4LMNAHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6951881-B2 (1-substituted-indol-3-yl) alkylidenehydrazinecarboximidamide derivatives as 5-hydroxytryptamine-6 ligands WYETH (US) 2005-10-04 US disclosed