SCHEMBL6494941

SCHEMBL6494941

NC(=O)CC1(c2ccc(-c3ccc(C(F)(F)F)cc3)cc2)CCCCC1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 6/20 0.60
SLC6A4 P31645 5/20 0.52
SLC6A2 P23975 2/20 0.52
HSD11B1 P28845 3/20 0.48
KIF11 P52732 5/20 0.43
P2RX7 Q99572 1/20 0.42
APP P05067 1/20 0.40
P2RY14 Q15391 1/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNB4 P30926 1/20 0.39
CHRNA3 P32297 1/20 0.39
CHRNA4 P43681 1/20 0.39
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6500186 0.99 SLC6A3 (0.57) SLC6A3SLC6A4SLC6A2HSD11B1KIF11
SCHEMBL17761315 0.94 SLC6A3 (0.62) SLC6A3SLC6A4SLC6A2HSD11B1P2RX7
SCHEMBL17761293 0.91 SLC6A3 (0.58) SLC6A3SLC6A4SLC6A2HSD11B1P2RX7
SCHEMBL17761224 0.88 SLC6A3 (0.53) SLC6A3SLC6A4SLC6A2HSD11B1KIF11
SCHEMBL6494518 0.84 HSD11B1 (0.68) SLC6A3SLC6A4SLC6A2HSD11B1
SCHEMBL6499750 0.82 HSD11B1 (0.65) SLC6A3SLC6A4SLC6A2HSD11B1
SCHEMBL6208426 0.82 SLC6A4 (0.64) SLC6A3SLC6A4SLC6A2HSD11B1
SCHEMBL6208549 0.81 SLC6A4 (0.61) SLC6A3SLC6A4SLC6A2HSD11B1
SCHEMBL2835624 0.81 SLC6A3 (0.90) SLC6A3SLC6A4SLC6A2
SCHEMBL15867331 0.80 SLC6A3 (0.62) SLC6A3SLC6A4SLC6A2HSD11B1P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050234096-A1 Tetrahydroisoquinoline derivatives BAYER HEALTHCARE AG (DE) 2005-10-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050234096-A1 Tetrahydroisoquinoline derivatives PPARD, PPARG, PPARA SLC6A3 3645/4885SLC6A4 3525/4885SLC6A2 3869/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.