SCHEMBL6499731

SCHEMBL6499731

O=C(NNNC(=S)c1ccc(Br)cc1)c1ccncc1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 6/20 0.57
ALDH1A1 P00352 5/20 0.53
LMNA P02545 3/20 0.53
PTGS1 P23219 1/20 0.52
PTGS2 P35354 1/20 0.52
CA1 P00915 3/20 0.51
CA9 Q16790 3/20 0.51
MAPT P10636 2/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
SMN1; SMN2 Q16637 3/20 0.47
UBE2N P61088 1/20 0.47
TP53 P04637 1/20 0.46
TLR7 Q9NYK1 1/20 0.46
POLB P06746 1/20 0.46
HPGD P15428 1/20 0.46
KDM4E B2RXH2 1/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6502042 0.85 CA1 (0.59) GAAALDH1A1LMNAPTGS2CA1
SCHEMBL6502761 0.85 KMT2A (0.54) GAAALDH1A1PTGS1PTGS2CA1
SCHEMBL6504612 0.84 GAA (0.57) GAAALDH1A1CA1CA9MEN1
SCHEMBL13492090 0.84 ALDH1A1 (0.76) GAAALDH1A1LMNAPTGS1PTGS2
SCHEMBL14527359 0.76 HDAC1 (0.68) GAAALDH1A1LMNAPTGS1PTGS2
SCHEMBL13481186 0.72 POLB (0.68) GAAALDH1A1LMNAMAPTMEN1
SCHEMBL1982518 0.72 POLB (0.68) GAAALDH1A1LMNAMAPTMEN1
SCHEMBL2992964 0.72 ALDH1A1 (1.00) GAAALDH1A1LMNAPTGS2CA1
SCHEMBL7553638 0.71 LMNA (0.50) GAAALDH1A1LMNAPTGS1PTGS2
SCHEMBL8387086 0.70 LMNA (0.76) GAAALDH1A1LMNAPTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6846933-B1 Antimycobacterial compounds and method for making the same THE BOARD OF TRUSTEES OF WELLESLEY COLLEGE (US) 2005-01-25 US disclosed
WO-2002043668-A2 ANTIMYCOBACTERIAL COMPOUNDS AND METHOD FOR MAKING THE SAME WELLESLEY COLLEGE (US) 2002-06-06 WO disclosed