SCHEMBL6501464

SCHEMBL6501464

CC(C)C(C(N)=O)c1nc(-c2ccccc2)cc(-c2ccccc2)n1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 10/20 0.50
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
ADORA3 P0DMS8 3/20 0.46
ADORA2A P29274 3/20 0.44
ADORA2B P29275 1/20 0.43
ALDH1A1 P00352 2/20 0.42
MAPT P10636 2/20 0.42
HPGD P15428 2/20 0.42
KDM4E B2RXH2 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
CYP2C19 P33261 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17563610 0.74 MEN1 (0.54) ADORA1MEN1KMT2AADORA3ADORA2A
SCHEMBL6501260 0.71 MEN1 (0.66) ADORA1MEN1KMT2AADORA3ADORA2A
SCHEMBL5475337 0.70 CYP2D6 (0.54) KMT2AKDM4ETSHR
SCHEMBL14749339 0.70 CYP2D6 (0.54) KMT2AKDM4ETSHR
SCHEMBL1483328 0.70 CYP2D6 (0.54) KMT2AKDM4ETSHR
SCHEMBL4651196 0.70 PDPK1 (0.39) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL7833643 0.69 FFAR2 (0.39) ALDH1A1KDM4ETSHR
SCHEMBL1733453 0.68 KDM4E (0.57) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL30938002 0.67 ADORA1 (0.61) ADORA1MEN1KMT2AADORA3ADORA2A
SCHEMBL22623614 0.67 MEN1 (0.44) ADORA1MEN1KMT2AADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033085-A1 PYRIMIDINES DERIVATIVES AS ADENOSINE RECEPTORS LIGANDS UNIVERSITEIT LEIDEN (NL) 2005-04-14 WO disclosed