SCHEMBL6501761

SCHEMBL6501761

CC(C)(C#N)NC(=O)C(CC1CCCCC1)NC1=NS(=O)(=O)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.46
CTSL P07711 5/20 0.41
CTSK P43235 3/20 0.41
CTSB P07858 3/20 0.41
MAPT P10636 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
TP53 P04637 1/20 0.36
HSD17B10 Q99714 1/20 0.36
FBP1 P09467 1/20 0.35
ALDH1A1 P00352 2/20 0.35
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6494159 0.86 CTSS (0.42) CTSSCTSLCTSKCTSB
SCHEMBL6528739 0.82 CTSS (0.54) CTSSCTSLCTSKCTSB
SCHEMBL5946020 0.81 KCNA3 (0.42) RXFP1SMN1; SMN2NPC1RAB9AFBP1
SCHEMBL5946029 0.81 KCNA3 (0.42) RXFP1SMN1; SMN2NPC1RAB9AFBP1
SCHEMBL5366946 0.79 CTSS (0.53) CTSSCTSLCTSKCTSB
SCHEMBL14383667 0.79 CTSS (0.53) CTSSCTSLCTSKCTSB
SCHEMBL14383668 0.76 CTSS (0.46) CTSSCTSLCTSKCTSB
SCHEMBL5368517 0.76 CTSS (0.46) CTSSCTSLCTSKCTSB
SCHEMBL5360338 0.75 CTSS (0.48) CTSSCTSL
SCHEMBL5372284 0.75 CTSS (0.48) CTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936606-B2 Cyanoamido-containing heterocyclic compounds useful as reversible inhibitors of cysteine proteases BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-08-30 US claimed
US-20040063679-A1 Compounds useful as reversible inhibitors of cysteine proteases BOEHRINGER INGELHEIM PHARMACEUTICALS INC. 2004-04-01 US claimed
US-6936606-B2 Cyanoamido-containing heterocyclic compounds useful as reversible inhibitors of cysteine proteases BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2005-08-30 US disclosed
US-20040063679-A1 Compounds useful as reversible inhibitors of cysteine proteases BOEHRINGER INGELHEIM PHARMACEUTICALS INC. 2004-04-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063679-A1 Compounds useful as reversible inhibitors of cysteine proteases CTSS, CTSK, CTSB CTSS 1/4885CTSL 8/4885CTSK 2/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.