SCHEMBL6502087

SCHEMBL6502087

CC(Br)c1ccc(CC(=O)O)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
HPGD P15428 2/20 0.53
HSD17B10 Q99714 2/20 0.53
CA2 P00918 1/20 0.52
CAMK2A Q9UQM7 1/20 0.52
AKR1B1 P15121 1/20 0.50
PTGS1 P23219 5/20 0.48
LMNA P02545 4/20 0.48
TSHR P16473 3/20 0.48
GAA P10253 2/20 0.48
ABCC4 O15439 1/20 0.48
HTT P42858 1/20 0.48
KLKB1 P03952 1/20 0.46
CTSB P07858 1/20 0.46
ANPEP P15144 1/20 0.44
ENPEP Q07075 1/20 0.44
FFAR1 O14842 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
PTGS2 P35354 4/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL909093 0.83 CA2 (0.56) ALDH1A1HPGDHSD17B10CA2CAMK2A
SCHEMBL27558460 0.82 HTT (0.40) ALDH1A1PTGS1LMNATSHRHTT
SCHEMBL10978746 0.82 CA2 (0.54) ALDH1A1HPGDHSD17B10CA2CAMK2A
SCHEMBL29248834 0.82 CA2 (0.54) ALDH1A1HPGDHSD17B10CA2CAMK2A
Hydrochloric Acid SCHEMBL2527629 0.82 CA2 (0.54) ALDH1A1HPGDHSD17B10CA2CAMK2A
SCHEMBL27649243 0.81 FFAR1 (0.55) ALDH1A1HSD17B10CA2LMNAFFAR1
SCHEMBL11795064 0.80 F2 (0.56) ALDH1A1HPGDHSD17B10CA2CAMK2A
SCHEMBL503594 0.80 CA2 (0.52) ALDH1A1HPGDHSD17B10CA2CAMK2A
SCHEMBL1061942 0.80 PTGS2 (0.67) CA2CAMK2AAKR1B1PTGS1LMNA
SCHEMBL29009922 0.80 CA2 (0.52) ALDH1A1HPGDHSD17B10CA2CAMK2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 33 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105531269-A \"inhibitors of nicotinamide phosphoribosyltransferase, compositions, products and uses thereof\ UNIV DEGLI STUDI DEL PIEMONTE ORIENTALE AMEDEO AVOGADRO 2016-04-27 CN disclosed
CN-105431422-A Isoindoline or isoquinoline compounds, process for their preparation and pharmaceutical compositions containing them SERVIER LAB 2016-03-23 CN disclosed
CN-105121423-A Novel 3- (4- (benzyloxy) phenyl) hex-4-ynoic acid derivative, method for preparing the same, and pharmaceutical composition for preventing and treating metabolic diseases comprising the same as an effective ingredient HYUNDAI PHARM CO LTD 2015-12-02 CN disclosed
CN-105073742-A Flap modulators JANSSEN PHARMACEUTICA NV 2015-11-18 CN disclosed
CN-102666567-B For the method and composition that the F-18 of the improvement of protein, peptide and other molecule marks IMMUNOMEDICS, INC. (US) 2015-08-26 CN disclosed
CN-104768932-A Heteroaryl inhibitors of PDE4 TETRA DISCOVERY PARTNERS LLC 2015-07-08 CN disclosed
CN-104693193-A Arylmethoxy isoindoline derivatives and compositions comprising and methods of using the same CELGENE CORP 2015-06-10 CN disclosed
CN-102822165-B Arylmethoxy isoindoline derivatives and compositions comprising and methods of using the same CELGENE CORP 2015-02-25 CN disclosed
CN-103068799-B Benzamide derivatives as HSP90 inhibitors and uses thereof CHROMA THERAPEUTICS LTD 2014-09-03 CN disclosed
CN-101402562-B Novel benzophenone derivatives or salts thereof TOYAMA CHEMICAL CO LTD 2013-07-31 CN disclosed
CN-101284808-A Compounds and methods for the inhibition of the expression of VCAM-1 ATHEROGENICS INC (US) 2008-10-15 CN disclosed
CN-101282949-A Azole and thiazole derivatives and their use ARGENTA DISCOVERY LTD (GB) 2008-10-08 CN disclosed
CN-101054345-A Novel bensophenone derivatives or salts thereof TOYAMA CHEMICAL CO LTD (JP) 2007-10-17 CN disclosed
CN-1914173-A Quinolines useful in treating cardiovascular disease WYETH CORP (US) 2007-02-14 CN disclosed
CN-1886376-A Pyridine compounds as dipeptidyl dipeptidase-IV inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2006-12-27 CN disclosed
CN-1878786-A Novel 17 beta-hydroxysteroid dehydrogenase type I inhibitors SOLVAY PHARM GMBH (DE) 2006-12-13 CN disclosed
CN-1602291-A Novel benzophenone derivative or salt thereof TOYAMA CHEMICAL CO LTD (JP) 2005-03-30 CN disclosed
WO-2005021496-A2 SYNTHESIS OF DERIVATIVES OF GINKGOLIDE C THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2005-03-10 WO disclosed
CN-1263522-A Compounds and methods for inhibiting VCAM-1 expression ATHEROGENICS INC (US) 2000-08-16 CN disclosed
CN-1202888-A Isoquinoline derivatives and isoquinoline combinatorial libraries TORREY PINES INST (US) 1998-12-23 CN disclosed