SCHEMBL6502485

SCHEMBL6502485

CC(=O)OCCCC(=O)Oc1ccc(CC(NC(=O)OCC(C)(C)C)C(C)C(=O)O)cc1C(C)=O

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.37
ITGAV P06756 1/20 0.37
ALOX15 P16050 2/20 0.35
CFD P00746 1/20 0.32
CTSK P43235 1/20 0.32
REN P00797 1/20 0.30
CTSD P07339 1/20 0.30
BACE1 P56817 1/20 0.30
PPARD Q03181 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6502488 0.85 ITGB3 (0.34) ITGB3ITGAVALOX15CFDCTSK
SCHEMBL14431790 0.84 ITGB3 (0.40) ITGB3ITGAVALOX15CTSK
SCHEMBL6502492 0.75 NPC1 (0.31) CTSK
SCHEMBL5206885 0.62 ITGB3 (0.44) ITGB3ITGAVCTSKBACE1
SCHEMBL14431256 0.62 ITGB3 (0.44) ITGB3ITGAVCTSKBACE1
SCHEMBL6495736 0.62 ITGB3 (0.44) ITGB3ITGAVALOX15CTSK
SCHEMBL1209402 0.62 ALOX15 (0.54) ITGB3ITGAVALOX15
SCHEMBL1212529 0.59 ALOX15 (0.40) ITGB3ITGAVALOX15
SCHEMBL1211298 0.59 ALOX15 (0.40) ITGB3ITGAVALOX15CFD
SCHEMBL10192477 0.59 P2RX1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849646-B1 Chromenone and chromanone derivatives as integrin inhibitors MERCK PATENT GMBH (DE) 2005-02-01 US disclosed