SCHEMBL6502486

SCHEMBL6502486

Cc1ccc2cc(N3CCC(C(=O)O)CC3)ccc2n1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 2/20 0.59
PDE3A Q14432 2/20 0.59
KDM4E B2RXH2 2/20 0.56
HSD17B10 Q99714 2/20 0.56
USP2 O75604 1/20 0.56
HPGD P15428 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
GAA P10253 1/20 0.48
TSHR P16473 1/20 0.48
CASP1 P29466 1/20 0.48
CASP7 P55210 1/20 0.48
NOTUM Q6P988 8/20 0.48
KMT2A Q03164 2/20 0.46
TP53 P04637 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
RHOA P61586 1/20 0.45
KDM2B Q8NHM5 1/20 0.45
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
AURKA O14965 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6500585 0.84 LGMN (0.61) PDE3BPDE3AKDM4EHSD17B10HPGD
SCHEMBL3864702 0.80 HRH3 (0.53) KDM4EHSD17B10USP2NPSR1GAA
Hydrochloric Acid SCHEMBL3863650 0.79 HRH3 (0.52) KDM4EHSD17B10USP2NPSR1GAA
SCHEMBL5799831 0.79 NOTUM (0.55) PDE3BPDE3AKDM4EHSD17B10USP2
SCHEMBL5800611 0.77 NOTUM (0.55) PDE3BPDE3AKDM4EHSD17B10USP2
SCHEMBL13683680 0.77 HRH3 (0.60) KDM4EHSD17B10USP2KMT2ATP53
SCHEMBL4891157 0.76 KDM4E (0.56) PDE3BPDE3AKDM4EHSD17B10USP2
SCHEMBL13683687 0.76 MAPT (0.42) PDE3BPDE3AKDM4EHSD17B10USP2
Hydrochloric Acid SCHEMBL3868535 0.76 HRH3 (0.59) KDM4EHSD17B10USP2KMT2ATP53
SCHEMBL6948711 0.76 HTR3E (0.57) KDM4EHSD17B10USP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005019200-A2 ARYL PIPERIDINE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed
WO-2005019200-A2 ARYL PIPERIDINE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-03-03 WO disclosed