SCHEMBL6502937

SCHEMBL6502937

CCOC(=O)C(=O)c1c(-c2ccc(Cl)cc2)c(-c2ccccc2)c2n1CC(C)(C)C2OC(C)=O

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 5/20 0.55
PTGS1 P23219 5/20 0.55
PTGS2 P35354 3/20 0.52
PTGES O14684 3/20 0.40
ALOX5AP P20292 1/20 0.40
HTT P42858 1/20 0.36
ATM Q13315 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CACNA1D Q01668 1/20 0.36
MAPT P10636 2/20 0.36
ALDH1A1 P00352 3/20 0.36
CYP19A1 P11511 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CYP1A2 P05177 1/20 0.33
HPGD P15428 1/20 0.33
XBP1 P17861 1/20 0.33
CYP2C19 P33261 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6495185 0.87 ALOX5 (0.51) ALOX5PTGS1PTGS2PTGESALOX5AP
SCHEMBL6499123 0.86 ALOX5 (0.50) ALOX5PTGS1PTGS2PTGESALOX5AP
SCHEMBL6503974 0.81 ALOX5 (0.81) ALOX5PTGS1PTGS2PTGESALOX5AP
SCHEMBL13844797 0.77 PTGES (0.61) ALOX5PTGS1PTGS2PTGESALOX5AP
SCHEMBL6495841 0.76 ALOX5 (0.74) ALOX5PTGS1PTGS2PTGESALOX5AP
SCHEMBL8397926 0.76 ALOX5 (0.45) ALOX5PTGS1PTGS2PTGESALOX5AP
SCHEMBL6496842 0.73 ALOX5 (0.47) ALOX5PTGS1PTGS2HTTATM
SCHEMBL6496837 0.73 ALOX5 (0.47) ALOX5PTGS1PTGS2HTTATM
SCHEMBL8394771 0.71 ALDH1A1 (0.39) ALOX5PTGS1PTGS2PTGESALOX5AP
SCHEMBL6505066 0.71 PTGES (0.44) ALOX5PTGS1PTGS2PTGESALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6878738-B1 Anti-inflammatory oxo derivatives and hydroxy derivatives of pyrrolizines, and their pharmaceutical use MERCKLE GMBH (DE) 2005-04-12 US disclosed