SCHEMBL6503058

SCHEMBL6503058

[CH2]NC(=O)c1ccc(OC)cc1OC

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.61
NPC1 O15118 6/20 0.58
RAB9A P51151 5/20 0.57
ALDH1A1 P00352 3/20 0.57
HPGD P15428 3/20 0.57
GAA P10253 2/20 0.57
KMT2A Q03164 2/20 0.57
PKM P14618 1/20 0.57
HTT P42858 1/20 0.57
HDAC3 O15379 1/20 0.57
HDAC1 Q13547 1/20 0.57
HDAC2 Q92769 1/20 0.57
MEN1 O00255 1/20 0.57
SMN1; SMN2 Q16637 2/20 0.55
MAPT P10636 2/20 0.55
MITF O75030 1/20 0.55
RAD52 P43351 1/20 0.53
ABCG2 Q9UNQ0 1/20 0.53
PRMT5 O14744 1/20 0.52
WDR77 Q9BQA1 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4154660 0.84 NPC1 (0.65) TP53NPC1RAB9AALDH1A1HPGD
SCHEMBL4939202 0.83 TP53 (0.66) TP53NPC1RAB9AALDH1A1HPGD
SCHEMBL6504797 0.82 TP53 (0.69) TP53NPC1RAB9AALDH1A1HPGD
SCHEMBL4900211 0.82 NPC1 (0.66) TP53NPC1RAB9AALDH1A1HPGD
SCHEMBL13761422 0.81 TP53 (0.68) TP53NPC1RAB9AALDH1A1HPGD
Methyl 2,4-Dimethoxybenzoate SCHEMBL645462 0.80 KMT2A (0.64) TP53NPC1RAB9AALDH1A1HPGD
SCHEMBL624926 0.80 NPC1 (0.64) TP53NPC1RAB9AALDH1A1HPGD
SCHEMBL10793237 0.80 TP53 (0.71) TP53NPC1RAB9AALDH1A1HPGD
SCHEMBL16149341 0.80 NPC1 (0.74) TP53NPC1RAB9AALDH1A1HPGD
SCHEMBL285924 0.80 NPC1 (0.79) TP53NPC1RAB9AALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed
US-6245779-B1 ANALGESICS; ANTIINFLAMMATORY AGENTS OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2001-06-12 US disclosed
CN-1262685-A Naphthyridine derivatives OTSUKA PHARMA CO LTD (JP) 2000-08-09 CN disclosed
EP-0997463-A1 NAPHTHYRIDINE DERIVATIVES OTSUKA PHARMACEUTICAL FACTORY, INC. (JP) 2000-05-03 EP disclosed