SCHEMBL6504440

SCHEMBL6504440

CC(C)Oc1ccc(C(=O)NCc2cc(CC(OC(C)C)C(=O)O)ccc2-c2ccsc2)c(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
ITGB1 P05556 2/20 0.36
ITGA4 P13612 2/20 0.36
PTGES O14684 3/20 0.35
PPARA Q07869 11/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
PPARG P37231 8/20 0.34
PPARD Q03181 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6495506 0.92 PPARA (0.38) PTGESPPARACD274PPARGPPARD
SCHEMBL6504030 0.92 PPARG (0.37) PPARAPPARGPPARD
SCHEMBL6502969 0.90 S1PR3 (0.38) EPHX2ITGB1ITGA4PPARAPPARG
SCHEMBL6502157 0.86 NR1H4 (0.37) EPHX2NR1H4ITGB1ITGA4PTGES
SCHEMBL6502348 0.85 EPHX2 (0.36) EPHX2NR1H4ITGB1ITGA4PPARA
SCHEMBL7685465 0.85 EPHX2 (0.36) EPHX2NR1H4ITGB1ITGA4PPARA
SCHEMBL6494327 0.85 EPHX2 (0.37) EPHX2NR1H4ITGB1ITGA4PPARA
SCHEMBL6505285 0.84 PPARA (0.43) EPHX2NR1H4PPARAPPARGPPARD
SCHEMBL6496963 0.82 TP53 (0.39) EPHX2NR1H4ITGB1ITGA4PPARA
SCHEMBL6503712 0.82 PPARA (0.50) PPARAPPARGPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed