SCHEMBL6504742

SCHEMBL6504742

CC(Br)Oc1cccc(N=C=O)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.38
TRPA1 O75762 1/20 0.38
MAPK1 P28482 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
HTR3E A5X5Y0 1/20 0.36
HTR3B O95264 1/20 0.36
HTR3A P46098 1/20 0.36
HTR3D Q70Z44 1/20 0.36
HTR3C Q8WXA8 1/20 0.36
TAAR1 Q96RJ0 1/20 0.35
TSHR P16473 2/20 0.35
ALDH1A1 P00352 1/20 0.35
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
ADRB2 P07550 1/20 0.32
MEN1 O00255 3/20 0.32
KMT2A Q03164 3/20 0.32
MAPT P10636 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6472016 0.87 RXRA (0.43) CYP3A4TRPA1MAPK1TDP1ALDH1A1
SCHEMBL1569276 0.80 DRD1 (0.46) MAPK1TDP1ALDH1A1MEN1KMT2A
SCHEMBL29541540 0.78 HTR3E (0.53) CYP3A4MAPK1TDP1HTR3EHTR3B
SCHEMBL23447 0.78 HTR3E (0.53) CYP3A4MAPK1TDP1HTR3EHTR3B
SCHEMBL11533412 0.77 MAPK1 (0.40) CYP3A4TRPA1MAPK1TDP1TSHR
SCHEMBL29808710 0.77 TDP1 (0.44) CYP3A4TRPA1MAPK1TDP1HTR3E
SCHEMBL5104173 0.77 TDP1 (0.44) CYP3A4TRPA1MAPK1TDP1HTR3E
SCHEMBL17911612 0.76 MTNR1A (0.40) TAAR1ALDH1A1RXRARXRBMEN1
SCHEMBL633675 0.76 MAPK1 (0.36) CYP3A4TRPA1MAPK1TDP1HTR3E
SCHEMBL7133728 0.75 CYP3A4 (0.44) CYP3A4TRPA1MAPK1TDP1HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005042495-A1 (BENZIMIDAZOL-2-YL)-PHENYL-PHENYL-UREA COMPOUNDS AND METHODS FOR INHIBITING HEPARANASE ACTIVITY IMCLONE SYSTEMS INCORPORATED (US) 2005-05-12 WO disclosed