SCHEMBL6505396

SCHEMBL6505396

COc1ncc(C=O)cc1CNC(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC13A5 Q86YT5 2/20 0.39
SLC13A2 Q13183 1/20 0.39
SLC13A3 Q8WWT9 1/20 0.39
PIK3CA P42336 1/20 0.38
ALDH1A1 P00352 5/20 0.36
TSHR P16473 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
POLB P06746 2/20 0.34
KDM4E B2RXH2 2/20 0.33
MAPK1 P28482 2/20 0.33
HPGD P15428 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
CFTR P13569 1/20 0.33
CHRM4 P08173 1/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15545023 0.85 SLC13A5 (0.40) SLC13A5SLC13A2SLC13A3PIK3CAALDH1A1
SCHEMBL3417608 0.81 SLC13A5 (0.40) SLC13A5SLC13A2SLC13A3ALDH1A1TSHR
SCHEMBL6498283 0.80 PPARG (0.41) ALDH1A1TSHRNPSR1KDM4EHPGD
SCHEMBL15545351 0.77 ATM (0.43) ALDH1A1SMN1; SMN2POLBMEN1NPC1
SCHEMBL15545354 0.77 ATM (0.43) ALDH1A1SMN1; SMN2POLBMEN1NPC1
SCHEMBL5034488 0.75 ALDH1A1 (0.51) ALDH1A1TSHRNPSR1SMN1; SMN2POLB
SCHEMBL6425131 0.75 MAOB (0.45) ALDH1A1NPSR1SMN1; SMN2NPC1RAB9A
SCHEMBL26101402 0.74 ALDH1A1 (0.45) PIK3CAALDH1A1TSHRSMN1; SMN2POLB
SCHEMBL26101902 0.74 NPC1 (0.43) SLC13A5SLC13A2SLC13A3PIK3CAALDH1A1
SCHEMBL15719149 0.73 FDPS (0.40) PIK3CAALDH1A1TSHRKDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6884821-B1 Carboxylic acid derivatives and drugs containing the same EISAI CO., LTD. (JP) 2005-04-26 US disclosed
EP-1216980-A1 CARBOXYLIC ACID DERIVATIVES AND DRUGS CONTAINING THE SAME Eisai Co., Ltd. (JP) 2002-06-26 EP disclosed