SCHEMBL6505891

SCHEMBL6505891

Cc1ccnc(C(N)c2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 2/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 1/20 0.42
NOS3 P29474 1/20 0.42
NOS1 P29475 1/20 0.42
KMT2A Q03164 1/20 0.42
UHRF1 Q96T88 1/20 0.41
CCR1 P32246 1/20 0.41
CCR5 P51681 1/20 0.41
CCR8 P51685 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
ROCK1 Q13464 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CYP1A2 P05177 1/20 0.37
KDR P35968 1/20 0.36
PLAU P00749 1/20 0.36
CRHR1 P34998 1/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28749349 0.79 NOS2 (0.50) NOS2KDM4EMEN1NOS3NOS1
SCHEMBL4428487 0.79 NOS2 (0.50) NOS2KDM4EMEN1NOS3NOS1
Hydrochloric Acid SCHEMBL31482081 0.77 NOS2 (0.48) NOS2KDM4EMEN1NOS3NOS1
SCHEMBL6513811 0.76 S1PR2 (0.48) NOS2KDM4ENOS3CCR1CCR5
SCHEMBL23619200 0.76 SLC6A2 (0.46) MEN1KMT2ASLC6A2SLC6A4SLC6A3
SCHEMBL2111803 0.75 SLC6A2 (0.63) KDM4ESLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL3384423 0.75 SLC6A2 (0.63) KDM4ESLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL6766141 0.75 SLC6A2 (0.63) KDM4ESLC6A2SLC6A4SLC6A3ALDH1A1
Hydrochloric Acid SCHEMBL7226415 0.73 SLC6A2 (0.61) KDM4ESLC6A2SLC6A4SLC6A3ALDH1A1
Hydrochloric Acid SCHEMBL4509965 0.73 SLC6A2 (0.61) KDM4ESLC6A2SLC6A4SLC6A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005023794-A2 COMPOUND LIBRARIES OF 4-CARBOXAMIDOPIPERIDINE DERIVATIVES BIOFOCUS PLC (GB) 2005-03-17 WO disclosed
WO-2004058755-A2 COMPOUND LIBRARIES OF IMIDAZO[1,5-A]PYRIDIN-3-YL DERIVATIVES AND RELATED HETEROBICYCLES FOR TARGETTING COMPOUNDS CAPABLE OF BINDING TO G-PROTEIN COUPLED RECEPTORS BIOFOCUS PLC (GB) 2004-07-15 WO disclosed